SCHEMBL22452004

SCHEMBL22452004

Cc1cccc2ccc(C(=O)OC(C)(C)C)nc12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.41
KDM4E B2RXH2 1/20 0.41
MMP2 P08253 1/20 0.40
PIM1 P11309 1/20 0.40
PFKFB3 Q16875 1/20 0.39
CYP1A2 P05177 1/20 0.39
AR P10275 1/20 0.38
ATM Q13315 3/20 0.37
ALDH1A1 P00352 2/20 0.37
HPGDS O60760 1/20 0.37
MAPT P10636 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
GABRP O00591 1/20 0.36
GABRD O14764 1/20 0.36
GABRA1 P14867 1/20 0.36
GABRB1 P18505 1/20 0.36
GABRG2 P18507 1/20 0.36
GABRB3 P28472 1/20 0.36
GABRA5 P31644 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23714070 0.83 CYP1A2 (0.47) KMT2AKDM4EMMP2PIM1CYP1A2
SCHEMBL22451969 0.82 CYP1A2 (0.41) KMT2AKDM4EPIM1CYP1A2HPGDS
SCHEMBL24454416 0.81 KDM4E (0.38) KMT2AKDM4EMMP2PIM1CYP1A2
SCHEMBL32315381 0.79 P2RX7 (0.50) KMT2AKDM4ECYP1A2ALDH1A1HPGDS
SCHEMBL946380 0.79 P2RX7 (0.50) KMT2AKDM4ECYP1A2ALDH1A1HPGDS
SCHEMBL1424052 0.77 KDM4E (0.66) KMT2AKDM4EMMP2PIM1PFKFB3
SCHEMBL4312684 0.76 MGAM (0.56) KMT2AKDM4EALDH1A1MAPTSMN1; SMN2
SCHEMBL6986429 0.76 MCHR1 (0.39) KMT2APIM1CYP1A2ALDH1A1SMN1; SMN2
SCHEMBL6984222 0.75 CYP1A2 (0.41) KDM4EMMP2PIM1CYP1A2ALDH1A1
SCHEMBL15724450 0.75 GRM6 (0.46) KMT2AKDM4EATMALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020186328-A1 CHELATORS AND METHODS OF MAKING AND USING SAME THE UNIVERSITY OF BRITISH COLUMBIA (CA) 2020-09-24 WO disclosed