SCHEMBL22452593

SCHEMBL22452593

CN1CCC(c2ccc(N(C)c3ccc(N)cc3)cc2)CC1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LSS P48449 1/20 0.49
QDPR P09417 2/20 0.45
SLC18A3 Q16572 2/20 0.44
HDAC3 O15379 1/20 0.42
HDAC4 P56524 1/20 0.42
HDAC1 Q13547 1/20 0.42
HDAC7 Q8WUI4 1/20 0.42
HDAC2 Q92769 1/20 0.42
HDAC10 Q969S8 1/20 0.42
HDAC11 Q96DB2 1/20 0.42
HDAC8 Q9BY41 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42
HDAC9 Q9UKV0 1/20 0.42
HDAC5 Q9UQL6 1/20 0.42
HTR1D P28221 1/20 0.40
HTR1B P28222 1/20 0.40
ALDH1A1 P00352 2/20 0.40
GFER P55789 2/20 0.40
KDM4E B2RXH2 1/20 0.40
GAA P10253 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL158531 0.88 QDPR (0.55) LSSQDPRSLC18A3HDAC3HDAC4
SCHEMBL22452582 0.83 CYP3A4 (0.43) SLC18A3ALDH1A1GFERESR2MAPK1
SCHEMBL22453195 0.81 SLC18A3 (0.44) SLC18A3HDAC1HDAC8HDAC6ALDH1A1
SCHEMBL14257946 0.81 SLC18A3 (0.58) LSSQDPRSLC18A3HDAC3HDAC4
SCHEMBL22452594 0.80 ESR2 (0.50) SLC18A3ALDH1A1GFERKDM4EMAPT
SCHEMBL328439 0.79 SLC18A3 (0.53) LSSQDPRSLC18A3HDAC3HDAC4
SCHEMBL22744420 0.78 LSS (0.44) LSSQDPRSLC18A3ESR2HSP90AA1
SCHEMBL14320804 0.78 SLC18A3 (0.46) LSSQDPRSLC18A3HTR1DHTR1B
SCHEMBL22453528 0.77 ESR2 (0.40) SLC18A3ALDH1A1GFERGAAESR2
SCHEMBL2056213 0.77 HTR2A (0.52) LSSQDPRALDH1A1KMT2AKDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020190774-A1 NOVEL SMALL MOLECULE INHIBITORS OF TEAD TRANSCRIPTION FACTORS THE GENERAL HOSPITAL CORPORATION (US) 2020-09-24 WO disclosed