SCHEMBL22452996

SCHEMBL22452996

CC(=N)c1cc(NC(=O)c2ccc(N)c(N)c2)ccc1N

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 2/20 0.50
KMT2A Q03164 4/20 0.45
MEN1 O00255 3/20 0.45
PKM P14618 2/20 0.45
KDM4E B2RXH2 1/20 0.45
NPC1 O15118 1/20 0.45
MAPT P10636 1/20 0.45
RAB9A P51151 1/20 0.45
HDAC1 Q13547 9/20 0.43
BRAF P15056 6/20 0.43
HDAC3 O15379 3/20 0.43
HDAC4 P56524 3/20 0.43
HDAC7 Q8WUI4 3/20 0.43
HDAC2 Q92769 3/20 0.43
HDAC10 Q969S8 3/20 0.43
HDAC11 Q96DB2 3/20 0.43
HDAC8 Q9BY41 3/20 0.43
HDAC6 Q9UBN7 3/20 0.43
HDAC9 Q9UKV0 3/20 0.43
HDAC5 Q9UQL6 3/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22453892 0.84 LRRK2 (0.55) LRRK2PKMNPC1RAB9AHDAC1
SCHEMBL11325167 0.83 KMT2A (0.55) KMT2AMEN1PKMKDM4ENPC1
SCHEMBL22453429 0.81 LRRK2 (0.42) LRRK2KMT2AMEN1PKMKDM4E
SCHEMBL22452944 0.80 LRRK2 (0.44) LRRK2KMT2AMEN1PKMKDM4E
SCHEMBL22453728 0.80 LRRK2 (0.44) LRRK2KMT2AMEN1PKMKDM4E
SCHEMBL22453889 0.78 LRRK2 (0.42) LRRK2KMT2AMEN1PKMKDM4E
SCHEMBL22453391 0.78 LRRK2 (0.44) LRRK2HDAC1BRAFHDAC3HDAC4
SCHEMBL1250383 0.78 RAB9A (0.63) KMT2AMEN1PKMNPC1MAPT
SCHEMBL22453342 0.78 LRRK2 (0.46) LRRK2HDAC1BRAFHDAC3HDAC4
SCHEMBL28308170 0.77 KMT2A (0.51) KMT2AMEN1PKMKDM4ENPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020191261-A1 INDAZOLES AS LRRK2 INHIBITORS E-SCAPE BIO, INC. (US) 2020-09-24 WO disclosed