SCHEMBL22453373

SCHEMBL22453373

CN(c1ccc(N)cn1)c1ccc(C2CCCCC2)cc1Cl

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PSMB5 P28074 1/20 0.38
BACE1 P56817 1/20 0.36
SLC6A2 P23975 4/20 0.34
SLC6A4 P31645 4/20 0.34
SLC6A3 Q01959 4/20 0.34
KCNH2 Q12809 2/20 0.34
CYP2D6 P10635 1/20 0.34
KDM4E B2RXH2 1/20 0.34
GLA P06280 1/20 0.34
HTT P42858 1/20 0.34
KMT2A Q03164 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
HIF1A Q16665 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
CHRNB2 P17787 1/20 0.32
CHRNA3 P32297 1/20 0.32
CHRNA7 P36544 1/20 0.32
PPARG P37231 2/20 0.32
PPARA Q07869 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22453567 0.80 PSMB5 (0.45) PSMB5BACE1KDM4EGLAHTT
SCHEMBL22452599 0.76 PSMB5 (0.46) PSMB5BACE1KDM4EGLAHTT
SCHEMBL22453370 0.72 BACE1 (0.36) PSMB5BACE1SLC6A2SLC6A4SLC6A3
SCHEMBL22405891 0.70 KDM4E (0.50) PSMB5BACE1KDM4EGLAHTT
SCHEMBL4062175 0.68 SMN1; SMN2 (0.49) SMN1; SMN2
SCHEMBL3786337 0.67 SLC6A2 (0.49) BACE1SLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL4061449 0.66 KDM4E (0.35) KCNH2KDM4EKMT2ASMN1; SMN2TDP1
SCHEMBL24666303 0.65 PSMB5 (0.44) PSMB5KCNH2KDM4EGLAHTT
SCHEMBL3781164 0.65 SLC6A2 (0.50) BACE1SLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL4029123 0.65 CYP2C19 (0.42) SLC6A2SLC6A4SLC6A3KCNH2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020190774-A1 NOVEL SMALL MOLECULE INHIBITORS OF TEAD TRANSCRIPTION FACTORS THE GENERAL HOSPITAL CORPORATION (US) 2020-09-24 WO disclosed