SCHEMBL22453370

SCHEMBL22453370

Cc1cc(N(C)c2ccc(C3CCCCC3)cc2Cl)ccc1N

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 1/20 0.36
S100B P04271 1/20 0.35
SLC6A2 P23975 4/20 0.35
SLC6A4 P31645 4/20 0.35
SLC6A3 Q01959 4/20 0.35
KCNH2 Q12809 2/20 0.35
CYP2D6 P10635 1/20 0.35
MAPK13 O15264 1/20 0.34
MAPK12 P53778 1/20 0.34
MAPK11 Q15759 1/20 0.34
MAPK14 Q16539 1/20 0.34
PSMB5 P28074 2/20 0.33
SLC18A3 Q16572 1/20 0.32
ADORA3 P0DMS8 1/20 0.31
HDAC1 Q13547 3/20 0.31
HDAC2 Q92769 3/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22452583 0.83 S100B (0.41) BACE1S100BPSMB5SLC18A3
SCHEMBL790114 0.77 BACE1 (0.47) BACE1HDAC1HDAC2
SCHEMBL25630463 0.75 ALDH1A1 (0.45) BACE1HDAC1HDAC2
SCHEMBL3786337 0.73 SLC6A2 (0.49) BACE1SLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL22453373 0.72 PSMB5 (0.38) BACE1SLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL3781164 0.72 SLC6A2 (0.50) BACE1SLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL22298075 0.72 CYP3A4 (0.45) BACE1S100BHDAC1HDAC2
SCHEMBL22453371 0.72 ALDH1A1 (0.40) BACE1SLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL20210026 0.70 SLC18A3 (0.41) BACE1PSMB5SLC18A3
SCHEMBL20210325 0.70 MAPT (0.39) BACE1PSMB5SLC18A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020190774-A1 NOVEL SMALL MOLECULE INHIBITORS OF TEAD TRANSCRIPTION FACTORS THE GENERAL HOSPITAL CORPORATION (US) 2020-09-24 WO disclosed