SCHEMBL22453473

SCHEMBL22453473

COC(=O)c1ccc(Nc2ccc(C3CCCCC3)cc2)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.56
SMN1; SMN2 Q16637 2/20 0.56
NPC1 O15118 2/20 0.56
EPHX2 P34913 1/20 0.56
HDAC8 Q9BY41 2/20 0.54
HDAC6 Q9UBN7 2/20 0.54
HDAC3 O15379 1/20 0.54
HDAC11 Q96DB2 1/20 0.54
DEGS1 O15121 1/20 0.54
MEN1 O00255 3/20 0.53
KMT2A Q03164 3/20 0.53
CYP2C19 P33261 2/20 0.53
CYP1A2 P05177 1/20 0.53
CYP2D6 P10635 1/20 0.53
CYP2C9 P11712 1/20 0.53
MAPT P10636 2/20 0.53
HDAC1 Q13547 1/20 0.51
HAO1 Q9UJM8 1/20 0.49
METAP2 P50579 1/20 0.47
HPGD P15428 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1790000 0.92 ALDH1A1 (0.59) ALDH1A1SMN1; SMN2NPC1EPHX2HDAC8
SCHEMBL2949436 0.92 ALDH1A1 (0.59) ALDH1A1SMN1; SMN2NPC1EPHX2HDAC8
SCHEMBL2944396 0.92 ALDH1A1 (0.59) ALDH1A1SMN1; SMN2NPC1EPHX2HDAC8
SCHEMBL31003794 0.91 ALDH1A1 (0.53) ALDH1A1SMN1; SMN2NPC1EPHX2HDAC8
SCHEMBL16684739 0.91 HDAC8 (0.61) ALDH1A1SMN1; SMN2NPC1EPHX2HDAC8
SCHEMBL15214831 0.88 ALDH1A1 (0.56) ALDH1A1SMN1; SMN2NPC1EPHX2HDAC8
SCHEMBL12488363 0.87 HDAC1 (0.56) ALDH1A1SMN1; SMN2NPC1EPHX2HDAC8
SCHEMBL21656481 0.85 ALDH1A1 (0.60) ALDH1A1SMN1; SMN2NPC1EPHX2HDAC8
SCHEMBL21656950 0.85 ALDH1A1 (0.60) ALDH1A1SMN1; SMN2NPC1EPHX2HDAC8
SCHEMBL7330029 0.85 HDAC8 (0.59) ALDH1A1SMN1; SMN2NPC1EPHX2HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020190774-A1 NOVEL SMALL MOLECULE INHIBITORS OF TEAD TRANSCRIPTION FACTORS THE GENERAL HOSPITAL CORPORATION (US) 2020-09-24 WO disclosed