SCHEMBL22454034

SCHEMBL22454034

CNc1cc(F)c(C(=O)Nc2ccc(N)c(C(C)=N)c2)c(F)c1C=N

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 2/20 0.40
HDAC1 Q13547 8/20 0.36
FADS1 O60427 2/20 0.35
BRAF P15056 5/20 0.35
CA1 P00915 3/20 0.34
CA2 P00918 3/20 0.34
CA9 Q16790 2/20 0.34
ALDH1A1 P00352 1/20 0.33
MAPK1 P28482 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
HDAC3 O15379 3/20 0.33
HDAC2 Q92769 3/20 0.33
NCOR2 Q9Y618 1/20 0.33
HDAC4 P56524 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22453761 0.91 FADS1 (0.35) LRRK2HDAC1FADS1BRAFCA1
SCHEMBL22454051 0.90 HDAC1 (0.36) LRRK2HDAC1FADS1BRAFCA1
SCHEMBL22453968 0.89 HDAC1 (0.34) LRRK2HDAC1FADS1BRAFCA1
SCHEMBL22453786 0.88 LRRK2 (0.36) LRRK2HDAC1FADS1BRAFCA1
SCHEMBL22454042 0.88 BRAF (0.35) HDAC1FADS1BRAFCA1CA2
SCHEMBL22453797 0.88 FADS1 (0.39) HDAC1FADS1ALDH1A1SMN1; SMN2KLK1
SCHEMBL22453911 0.88 HDAC1 (0.40) HDAC1FADS1BRAFALDH1A1MAPK1
SCHEMBL22453587 0.87 CYP3A4 (0.33) HDAC1FADS1BRAFCA1CA2
SCHEMBL22454069 0.87 HDAC1 (0.33) LRRK2HDAC1FADS1BRAFCA1
SCHEMBL22453923 0.87 HDAC1 (0.32) LRRK2HDAC1FADS1BRAFCA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020191261-A1 INDAZOLES AS LRRK2 INHIBITORS E-SCAPE BIO, INC. (US) 2020-09-24 WO disclosed