SCHEMBL22474472

SCHEMBL22474472

c1ccc2c(c1)CC1CCCC(Cc3ccccc3O1)O2

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 2/20 0.42
CHRM4 P08173 2/20 0.42
CHRM5 P08912 2/20 0.42
CHRM1 P11229 2/20 0.42
CHRM3 P20309 2/20 0.42
HPGD P15428 1/20 0.42
TSHR P16473 1/20 0.42
MAOA P21397 7/20 0.39
MAOB P27338 7/20 0.39
AOC2 O75106 5/20 0.39
DAO P14920 1/20 0.39
NISCH Q9Y2I1 1/20 0.37
HRH3 Q9Y5N1 1/20 0.36
ESR1 P03372 1/20 0.35
ESR2 Q92731 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29935960 0.76 MAOB (0.42) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL5722720 0.76 MAOB (0.42) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL14837286 0.72 TSHR (0.39) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL17891950 0.71 CHRM2 (0.58) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL10698516 0.71 MAOB (0.39) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL1579371 0.71 CHRM2 (0.50) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL7424079 0.71 CHRM2 (0.54) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL22474527 0.70 DRD2 (0.43) MAOB
SCHEMBL8470150 0.70 BRD4 (0.50) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL20801116 0.70 CHRM2 (0.45) CHRM2CHRM4CHRM5CHRM1CHRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2876108-B1 COMPOUNDS OF CHIRAL AROMATIC SPIROKETAL DIPHOSPHINE LIGANDS, PREPARATION METHODS AND USES THEREOF SHANGHAI INST ORGANIC CHEMISTRY CAS (CN) 2020-09-30 EP disclosed