SCHEMBL22474643

SCHEMBL22474643

C=C(/C=C(CCC(=O)OCC)\C(=C/C)C(=O)OC)OC

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.35
MGAM O43451 1/20 0.35
SI P14410 1/20 0.35
MGAM2 Q2M2H8 1/20 0.35
NPSR1 Q6W5P4 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP4F2 P78329 2/20 0.32
CYP4A11 Q02928 2/20 0.32
NR1I2 O75469 1/20 0.31
PGR P06401 1/20 0.31
ADORA3 P0DMS8 1/20 0.31
PTGS2 P35354 1/20 0.31
PDE4D Q08499 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
POLB P06746 2/20 0.31
TSHR P16473 2/20 0.31
LMNA P02545 1/20 0.31
ALDH1A1 P00352 4/20 0.30
CYP2D6 P10635 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL280330 0.75 TSHR (0.48) GAAMGAMSIMGAM2L3MBTL1
SCHEMBL17108458 0.69 NPSR1 (0.54) GAAMGAMSIMGAM2NPSR1
SCHEMBL19296253 0.69 NPSR1 (0.54) GAAMGAMSIMGAM2NPSR1
Ethylene Glycol SCHEMBL2782790 0.68 TSHR (0.48) GAAMGAMSIMGAM2CYP1A2
SCHEMBL28244616 0.66 CYP1A2 (0.42) GAAMGAMSIMGAM2CYP1A2
SCHEMBL1981808 0.66 TSHR (0.68) GAAMGAMSIMGAM2CYP1A2
Succinic Acid Diethyl Ester SCHEMBL28083672 0.66 GAA (0.60) GAAMGAMSIMGAM2CYP1A2
SCHEMBL1911255 0.66 CYP1A2 (0.45) GAAMGAMSIMGAM2CYP1A2
Succinic Acid Diethyl Ester SCHEMBL22780 0.66 GAA (0.67) GAAMGAMSIMGAM2CYP1A2
Succinic Acid Diethyl Ester SCHEMBL27768067 0.66 GAA (0.67) GAAMGAMSIMGAM2CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2880028-B1 ANTIDIABETIC TRICYCLIC COMPOUNDS MERCK SHARP & DOHME (US) 2020-09-30 EP disclosed