SCHEMBL22482091

SCHEMBL22482091

CC(=O)NCCC1(O)CC(F)(F)C1

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.40
MAPK1 P28482 1/20 0.40
HIF1A Q16665 1/20 0.40
TSHR P16473 2/20 0.38
ALDH1A1 P00352 1/20 0.36
PAOX Q6QHF9 3/20 0.34
ADRA1A P35348 1/20 0.33
NQO2 P16083 1/20 0.33
KMT2A Q03164 1/20 0.33
NPSR1 Q6W5P4 1/20 0.32
F13A1 P00488 1/20 0.31
MTNR1A P48039 1/20 0.30
MTNR1B P49286 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24333752 0.81 KMT2A (0.36) MAPK1TSHRKMT2A
SCHEMBL22482075 0.79 KDM4E (0.46) KDM4EMAPK1HIF1ATSHRALDH1A1
SCHEMBL18629003 0.74 KDM4E (0.41) KDM4EMAPK1HIF1ATSHRALDH1A1
SCHEMBL22482085 0.69 KDM4E (0.40) KDM4EMAPK1HIF1ATSHRALDH1A1
SCHEMBL24618588 0.69 KDM4E (0.40) KDM4EMAPK1HIF1ATSHRALDH1A1
SCHEMBL22482095 0.68 OPRM1 (0.41) KDM4EMAPK1HIF1ATSHRALDH1A1
SCHEMBL22482084 0.68 KDM4E (0.54) KDM4EMAPK1HIF1ATSHRALDH1A1
SCHEMBL22434968 0.67 KDM4E (0.46) KDM4EMAPK1HIF1ATSHRALDH1A1
SCHEMBL25608117 0.65 KDM4E (0.44) KDM4EMAPK1HIF1ATSHRALDH1A1
SCHEMBL25106399 0.65 NPSR1 (0.41) KDM4EMAPK1HIF1ATSHRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020198583-A1 BICYCLIC JAK INHIBITORS AND USES THEREOF INSILICO MEDICINE IP LIMITED (CN) 2020-10-01 WO disclosed