SCHEMBL22482286

SCHEMBL22482286

CC(C)(C)OC(=O)N1CCc2snc(C(=O)CNCCC(F)(F)F)c2C1

nearest known ligand 0.37

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 2/20 0.37
TGM2 P21980 1/20 0.35
PRKCI P41743 1/20 0.34
GRAMD1A Q96CP6 1/20 0.34
SCN9A Q15858 1/20 0.34
MKNK1 Q9BUB5 7/20 0.33
KDM4E B2RXH2 1/20 0.33
MAPT P10636 1/20 0.33
ESR2 Q92731 1/20 0.33
NR1H2 P55055 1/20 0.33
P2RX3 P56373 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22482230 0.86 ADORA1 (0.39) ADORA1TGM2PRKCIGRAMD1ASCN9A
SCHEMBL22482233 0.78 ADORA1 (0.52) ADORA1GRAMD1ASCN9AMKNK1KDM4E
SCHEMBL22482028 0.75 ADORA1 (0.56) ADORA1KDM4EMAPTESR2NR1H2
SCHEMBL10413878 0.73 ADORA1 (0.48) ADORA1GRAMD1ASCN9AMKNK1KDM4E
SCHEMBL22482231 0.69 ADORA1 (0.45) ADORA1MKNK1KDM4EMAPTESR2
SCHEMBL22482006 0.69 RBP4 (0.41)
SCHEMBL22481978 0.69 HSP90AA1 (0.45) MAPT
SCHEMBL6424372 0.63 ADORA1 (0.53) ADORA1GRAMD1AMKNK1KDM4EMAPT
SCHEMBL7989573 0.62 ADORA1 (0.47) ADORA1MKNK1KDM4EMAPTESR2
SCHEMBL10413882 0.62 F12 (0.32) ADORA1KDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020198583-A1 BICYCLIC JAK INHIBITORS AND USES THEREOF INSILICO MEDICINE IP LIMITED (CN) 2020-10-01 WO disclosed