SCHEMBL22497580

SCHEMBL22497580

Nc1cccc(C(=O)Nc2c(Br)cc(C(F)(C(F)(F)F)C(F)(F)F)cc2I)c1F

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 5/20 0.40
P2RX1 P51575 2/20 0.39
RXFP1 Q9HBX9 3/20 0.36
SMN1; SMN2 Q16637 3/20 0.34
NPC1 O15118 3/20 0.34
RAB9A P51151 3/20 0.34
KDM4E B2RXH2 1/20 0.34
CASP3 P42574 1/20 0.34
SENP8 Q96LD8 1/20 0.34
HSD17B10 Q99714 1/20 0.34
SENP7 Q9BQF6 1/20 0.34
SENP6 Q9GZR1 1/20 0.34
CRBN Q96SW2 1/20 0.34
F2R P25116 1/20 0.33
MEN1 O00255 1/20 0.33
OPRK1 P41145 1/20 0.33
HTT P42858 1/20 0.33
KMT2A Q03164 1/20 0.33
FADS1 O60427 1/20 0.33
P2RX7 Q99572 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1767173 0.92 PTGS1 (0.43) PTGS1P2RX1RXFP1SMN1; SMN2NPC1
SCHEMBL1766487 0.92 PTGS1 (0.43) PTGS1P2RX1RXFP1NPC1RAB9A
SCHEMBL31175820 0.88 PTGS1 (0.40) PTGS1P2RX1RXFP1SMN1; SMN2NPC1
SCHEMBL29549892 0.87 PTGS1 (0.42) PTGS1P2RX1RXFP1SMN1; SMN2NPC1
SCHEMBL1767085 0.87 PTGS1 (0.42) PTGS1P2RX1RXFP1SMN1; SMN2NPC1
SCHEMBL29615074 0.87 PTGS1 (0.42) PTGS1P2RX1RXFP1SMN1; SMN2CRBN
SCHEMBL16155678 0.87 FADS1 (0.40) PTGS1P2RX1RXFP1SMN1; SMN2NPC1
SCHEMBL1766505 0.87 PTGS1 (0.42) PTGS1P2RX1RXFP1SMN1; SMN2CRBN
SCHEMBL1766729 0.87 PTGS1 (0.41) PTGS1P2RX1RXFP1SMN1; SMN2KDM4E
SCHEMBL29161215 0.86 RXFP1 (0.40) RXFP1SMN1; SMN2NPC1RAB9AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117342978-A Cyanomethylation method of amine 沈阳化工大学 2024-01-05 CN disclosed
WO-2021139370-A1 AMIDE COMPOUND AND APPLICATION THEREOF 沈阳化工大学 2021-07-15 WO disclosed
WO-2021139370-A1 AMIDE COMPOUND AND APPLICATION THEREOF 沈阳化工大学 2021-07-15 WO disclosed
WO-2021036966-A1 BISAMIDE COMPOUND AND APPLICATION THEREOF 沈阳化工大学 2021-03-04 WO disclosed
WO-2021036966-A1 BISAMIDE COMPOUND AND APPLICATION THEREOF 沈阳化工大学 2021-03-04 WO disclosed
WO-2021036965-A1 ISOPHTHALAMIDE COMPOUND AND USE THEREOF 沈阳化工大学 2021-03-04 WO disclosed
WO-2020200290-A1 META-DIAMIDE COMPOUND AND APPLICATION THEREOF 沈阳化工大学 2020-10-08 WO disclosed