SCHEMBL22497614

SCHEMBL22497614

CPC.Nc1ccc2ccccc2c1Oc1c(N)ccc2ccccc12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.43
TSHR P16473 4/20 0.43
HSD17B10 Q99714 4/20 0.43
CYP3A4 P08684 2/20 0.43
HPGD P15428 2/20 0.43
KEAP1 Q14145 1/20 0.43
HPRT1 P00492 2/20 0.41
CYP2A6 P11509 3/20 0.41
TDP1 Q9NUW8 1/20 0.41
IDO1 P14902 1/20 0.37
MAPT P10636 1/20 0.37
CYP1A2 P05177 1/20 0.36
EP300 Q09472 1/20 0.36
KAT8 Q9H7Z6 1/20 0.36
NCEH1 Q6PIU2 1/20 0.36
HIF1A Q16665 2/20 0.35
CYP1B1 Q16678 1/20 0.35
F12 P00748 1/20 0.34
PLAU P00749 1/20 0.34
NCF1 P14598 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5623654 0.92 ALDH1A1 (0.50) ALDH1A1TSHRHSD17B10CYP3A4HPGD
Hydrochloric Acid SCHEMBL5967545 0.90 ALDH1A1 (0.48) ALDH1A1TSHRHSD17B10CYP3A4HPGD
SCHEMBL27976243 0.81 MAPT (0.50) ALDH1A1TSHRHSD17B10CYP3A4HPGD
Pyrimidine SCHEMBL5624365 0.80 ALDH1A1 (0.39) ALDH1A1TSHRHSD17B10CYP3A4HPGD
SCHEMBL358051 0.80 ALDH1A1 (0.50) ALDH1A1TSHRHSD17B10CYP3A4HPGD
SCHEMBL1806270 0.76 SLC2A1 (0.46) ALDH1A1TSHRHSD17B10CYP3A4HPGD
SCHEMBL31610446 0.76 ALDH1A1 (0.42) ALDH1A1TSHRHSD17B10CYP3A4HPGD
SCHEMBL3635012 0.75 CYP2A6 (0.58) ALDH1A1TSHRHSD17B10CYP3A4HPGD
SCHEMBL4688821 0.74 ALDH1A1 (0.47) ALDH1A1TSHRHSD17B10CYP3A4HPGD
SCHEMBL23174989 0.72 ALDH1A1 (0.42) ALDH1A1TSHRHSD17B10CYP3A4HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113677680-B EGFR inhibitor, composition and application thereof 贝达药业股份有限公司 2024-05-10 CN disclosed
CN-116891502-A EGFR degrading agent 上海齐鲁制药研究中心有限公司 2023-10-17 CN disclosed
CN-113166103-B EGFR inhibitor and application thereof 江苏先声药业有限公司 2022-12-16 CN disclosed
CN-113677680-A EGFR inhibitor and composition and application thereof 贝达药业股份有限公司 2021-11-19 CN disclosed
CN-113166103-A EGFR inhibitor and application thereof 江苏先声药业有限公司 2021-07-23 CN disclosed
WO-2020200191-A1 EGFR INHIBITORS, COMPOSITIONS AND METHODS THERE OF BETTA PHARMACEUTICALS CO., LTD (CN) 2020-10-08 WO disclosed