SCHEMBL22499861

SCHEMBL22499861

CC(C)(C)N(C(=O)O)[C@H]1CCN(c2ccc(C(F)(F)F)nc2)C1

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 1/20 0.48
CCNC P24863 1/20 0.48
CDK8 P49336 1/20 0.48
CYP3A4 P08684 2/20 0.47
CHRM4 P08173 4/20 0.44
PPARD Q03181 1/20 0.43
PPARA Q07869 1/20 0.43
USP30 Q70CQ3 1/20 0.41
NR1H2 P55055 2/20 0.41
NR1H3 Q13133 1/20 0.41
NOTUM Q6P988 1/20 0.41
LCAT P04180 2/20 0.40
MCHR1 Q99705 2/20 0.40
DHFR P00374 1/20 0.40
CHRM2 P08172 1/20 0.39
KCNH2 Q12809 1/20 0.39
GPR119 Q8TDV5 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22499863 1.00 HRH3 (0.48) HRH3CCNCCDK8CYP3A4CHRM4
SCHEMBL22499830 0.86 SLC6A9 (0.41) HRH3CHRM4PPARDPPARANOTUM
SCHEMBL22499829 0.86 SLC6A9 (0.41) HRH3CHRM4PPARDPPARANOTUM
SCHEMBL16398200 0.85 MCHR1 (0.40) CCNCCDK8NOTUMMCHR1
SCHEMBL22499979 0.84 ACACB (0.48) HRH3CHRM4NOTUMCHRM2
SCHEMBL22499980 0.84 ACACB (0.48) HRH3CHRM4NOTUMCHRM2
SCHEMBL16398478 0.83 MAPT (0.51) MCHR1
SCHEMBL16398474 0.83 MAPT (0.51) MCHR1
SCHEMBL1261496 0.83 NOTUM (0.60) CYP3A4CHRM4PPARDPPARANOTUM
SCHEMBL22499825 0.81 SLC6A9 (0.43) HRH3LCAT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020203610-A1 USE OF T-TYPE CALCIUM CHANNEL BLOCKER FOR TREATING RHEUMATOID ARTHRITIS 日本ケミファ株式会社 2020-10-08 WO disclosed