SCHEMBL22504153

SCHEMBL22504153

CC(=O)NS(=O)(=O)N1CCc2cc(Br)ccc2C1

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 4/20 0.53
ESR2 Q92731 3/20 0.47
ESR1 P03372 2/20 0.47
ACACB O00763 1/20 0.47
HSD17B3 P37058 3/20 0.46
CARM1 Q86X55 1/20 0.43
ABHD6 Q9BV23 1/20 0.42
HDAC6 Q9UBN7 2/20 0.41
PPARG P37231 2/20 0.39
PPARD Q03181 2/20 0.39
PPARA Q07869 2/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
OPRK1 P41145 2/20 0.39
OPRM1 P35372 1/20 0.38
OPRD1 P41143 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3175986 0.79 ESR2 (0.68) AKR1C3ESR2ESR1HSD17B3CARM1
SCHEMBL38665856 0.77 AKR1C3 (0.55) AKR1C3ESR2ESR1ACACBHSD17B3
SCHEMBL22504152 0.77 AKR1C3 (0.55) AKR1C3ESR2ESR1HSD17B3CARM1
SCHEMBL38666129 0.76 AKR1C3 (0.43) AKR1C3ESR2ESR1ACACBHSD17B3
SCHEMBL38666463 0.75 AKR1C3 (0.42) AKR1C3ESR2ESR1ACACBHSD17B3
SCHEMBL38664468 0.73 NMT1 (0.53) AKR1C3ESR2ESR1
SCHEMBL38666485 0.73 AKR1C3 (0.43) AKR1C3ESR2ESR1HSD17B3CARM1
SCHEMBL38666419 0.73 AKR1C3 (0.43) AKR1C3ESR2ESR1HSD17B3CARM1
SCHEMBL1265874 0.73 ESR1 (0.59) AKR1C3ESR2ESR1HSD17B3CARM1
SCHEMBL2185429 0.73 NOTUM (0.63) ESR2ESR1ACACBHSD17B3CARM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020200317-A1 TETRAHYDROISOQUINOLINE SULFONYLAMIDE DERIVATIVE, PREPARATION METHOD THEREFOR AND MEDICAL USE THEREOF 上海海雁医药科技有限公司 2020-10-08 WO disclosed