SCHEMBL22504152

SCHEMBL22504152

NS(=O)(=O)N1CCc2cc(Br)ccc2C1

nearest known ligand 0.55

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 2/20 0.55
CA7 P43166 1/20 0.54
ESR2 Q92731 4/20 0.49
ESR1 P03372 3/20 0.49
ENPP1 P22413 1/20 0.46
HSD17B3 P37058 3/20 0.43
ABHD6 Q9BV23 1/20 0.43
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
TSHR P16473 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
CARM1 Q86X55 1/20 0.41
HDAC6 Q9UBN7 1/20 0.39
ASIC3 Q9UHC3 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL38665856 0.87 AKR1C3 (0.55) AKR1C3CA7ESR2ESR1HSD17B3
SCHEMBL3175986 0.85 ESR2 (0.68) AKR1C3CA7ESR2ESR1HSD17B3
SCHEMBL20910236 0.80 CA7 (0.58) AKR1C3CA7ESR2ESR1ENPP1
SCHEMBL1265874 0.79 ESR1 (0.59) AKR1C3CA7ESR2ESR1HSD17B3
SCHEMBL20046985 0.78 AKR1C3 (0.60) AKR1C3ESR2MEN1KMT2AHDAC6
SCHEMBL2590065 0.78 AKR1C3 (0.60) AKR1C3ESR2MEN1KMT2AHDAC6
SCHEMBL22504153 0.77 AKR1C3 (0.53) AKR1C3ESR2ESR1HSD17B3ABHD6
SCHEMBL19748783 0.77 OPRK1 (0.54) AKR1C3ESR2ESR1MEN1KMT2A
SCHEMBL1033548 0.77 KMT2A (0.66) AKR1C3CA7MEN1KMT2ATSHR
SCHEMBL29843194 0.77 KMT2A (0.66) AKR1C3CA7MEN1KMT2ATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020200317-A1 TETRAHYDROISOQUINOLINE SULFONYLAMIDE DERIVATIVE, PREPARATION METHOD THEREFOR AND MEDICAL USE THEREOF 上海海雁医药科技有限公司 2020-10-08 WO disclosed