SCHEMBL2250806

SCHEMBL2250806

COc1ccc2nccc(CC[C@]3(O)CC[C@@](O)(CNc4ccc5c(c4)OCCO5)CC3)c2n1

nearest known ligand 0.49

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 13/20 0.49
SLC2A1 P11166 1/20 0.38
CDK4 P11802 1/20 0.37
CDK2 P24941 1/20 0.37
GSK3B P49841 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2250813 1.00 KCNH2 (0.49) KCNH2SLC2A1CDK4CDK2GSK3B
SCHEMBL2248805 0.85 KCNH2 (0.55) KCNH2
SCHEMBL3251533 0.85 KCNH2 (0.49) KCNH2
SCHEMBL1147947 0.84 KCNH2 (0.52) KCNH2
SCHEMBL1147476 0.84 KCNH2 (0.52) KCNH2
SCHEMBL3687649 0.80 KCNH2 (0.74) KCNH2
SCHEMBL3687651 0.80 KCNH2 (0.74) KCNH2
SCHEMBL3687657 0.80 KCNH2 (0.74) KCNH2
SCHEMBL2250560 0.80 KCNH2 (0.43) KCNH2SLC2A1
SCHEMBL4137510 0.80 KCNH2 (0.43) KCNH2SLC2A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7999115-B2 Spiro antibiotic derivatives ACTELION PHARMACEUTICAL LTD. (SE) 2011-08-16 US disclosed