SCHEMBL225149

SCHEMBL225149

Nc1ccc(-c2cccnc2)cc1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 5/20 0.68
CYP3A4 P08684 4/20 0.68
ALDH1A1 P00352 3/20 0.68
CYP1A2 P05177 1/20 0.68
MKNK1 Q9BUB5 5/20 0.64
MKNK2 Q9HBH9 5/20 0.64
MEN1 O00255 1/20 0.64
PSIP1 O75475 1/20 0.64
AXL P30530 1/20 0.64
CA12 O43570 1/20 0.58
CA1 P00915 1/20 0.58
CA2 P00918 1/20 0.58
CA9 Q16790 1/20 0.58
CYP11B2 P19099 2/20 0.57
KIF11 P52732 1/20 0.57
HSD17B10 Q99714 2/20 0.54
TDP1 Q9NUW8 2/20 0.54
TAAR1 Q96RJ0 1/20 0.54
MAPT P10636 2/20 0.52
HTT P42858 2/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29818169 1.00 CYP2A6 (0.68) CYP2A6CYP3A4ALDH1A1CYP1A2MKNK1
SCHEMBL18745788 1.00 CYP2A6 (0.68) CYP2A6CYP3A4ALDH1A1CYP1A2MKNK1
SCHEMBL18745701 0.92 MKNK1 (0.72) CYP2A6CYP3A4ALDH1A1CYP1A2MKNK1
SCHEMBL18745798 0.92 MKNK1 (0.63) CYP2A6CYP3A4ALDH1A1CYP1A2MKNK1
SCHEMBL11170593 0.89 AXL (0.86) CYP2A6CYP3A4ALDH1A1CYP1A2MKNK1
SCHEMBL28191166 0.89 CYP2A6 (0.54) CYP2A6CYP3A4ALDH1A1CYP1A2MKNK1
SCHEMBL24534338 0.88 CYP2A6 (0.88) CYP2A6CYP3A4ALDH1A1CYP1A2MKNK1
SCHEMBL29360677 0.88 CYP2A6 (0.88) CYP2A6CYP3A4ALDH1A1CYP1A2MKNK1
SCHEMBL13907273 0.88 CYP2A6 (0.88) CYP2A6CYP3A4ALDH1A1CYP1A2MKNK1
SCHEMBL18745763 0.87 CYP2A6 (0.57) CYP2A6CYP3A4ALDH1A1CYP1A2MKNK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 331 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109134351-B Synthesis method of S-3- (4-aminophenyl) piperidine 武汉理工大学 2022-03-11 CN claimed
US-20210145818-A1 COMPOSITIONS INFUSED WITH NICOTINE COMPOUNDS AND METHODS OF USE THEREOF Poviva Corp. 2021-05-20 US claimed
EP-3781163-A1 COMPOSITIONS INFUSED WITH NICOTINE COMPOUNDS AND METHODS OF USE THEREOF Poviva Corp. (US) 2021-02-24 EP claimed
EP-3284467-B1 NICOTINE-CONTAINING PHARMACEUTICAL COMPOSITIONS NICONOVUM USA INC (US) 2019-10-30 EP claimed
WO-2019202396-A1 COMPOSITIONS INFUSED WITH NICOTINE COMPOUNDS AND METHODS OF USE THEREOF POVIVA TEA, LLC (US) 2019-10-24 WO claimed
CN-109134351-A S-3-(4- aminophenyl) piperidines synthetic method 武汉理工大学 2019-01-04 CN claimed
US-9937168-B2 Nicotine-containing pharmaceutical compositions NICONOVUM USA, INC. (US) 2018-04-10 US claimed
EP-3284467-A1 NICOTINE-CONTAINING PHARMACEUTICAL COMPOSITIONS Niconovum USA, Inc. (US) 2018-02-21 EP claimed
EP-2566476-B1 NICOTINE-CONTAINING PHARMACEUTICAL COMPOSITIONS NICONOVUM USA INC (US) 2017-11-22 EP claimed
EP-2050749-B1 PYRIMIDINE DERIVATIVE AS PI3K INHIBITOR AND USE THEREOF CHUGAI PHARMACEUTICAL CO LTD (JP) 2017-11-22 EP claimed
CN-102892418-A Nicotine-containing pharmaceutical compositions NICONOVUM USA INC 2013-01-23 CN claimed
US-20100069629-A1 PYRIMIDINE DERIVATIVES AS PI3K INHIBITOR AND USE THEREOF CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2010-03-18 US claimed
WO-2009125923-A2 NOVEL INDOL CARBOXYLIC ACID BISPYRIDYL CARBOXAMIDE DERIVATIVES, PHARMACEUTICALLY ACCEPTABLE SALT THEREOF, PREPARATION METHOD AND COMPOSITION CONTAINING THE SAME AS AN ACTIVE INGREDIENT KOREA RESERACH INSTITUTE OF CHEMICAL TECHNOLOGY (KR) 2009-10-15 WO claimed
US-20090258876-A1 NOVEL INDOL CARBOXYLIC ACID BISPYRIDYL CARBOXAMIDE DERIVATIVES, PHARMACEUTICALLY ACCEPTABLE SALT THEREOF, PREPARATION METHOD AND COMPOSITION CONTAINING THE SAME AS AN ACTIVE INGREDIENT KOREA RESEARCH INSTITUTE OF CHEMICAL TECHNOLOGY (KR) 2009-10-15 US claimed
EP-2108649-A1 Novel indol carboxylic acid bispyridyl carboxamide derivatives as 5-HT2c receptor antagonists Korea Research Institute of Chemical Technology (KR) 2009-10-14 EP claimed
EP-2050749-A1 PYRIMIDINE DERIVATIVE AS PI3K INHIBITOR AND USE THEREOF CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2009-04-22 EP claimed
US-20080207694-A1 Hydroxamates as Histone Deacetylase Inhibitors and Pharmaceutical Formulations Containing Them ROSSI CRISTINA 2008-08-28 US claimed
EP-1868997-A1 HYDROXAMATES AS HISTONE DEACETYLASE INHIBITORS AND PHARMACEUTICAL FORMULATIONS CONTAINING THEM Menarini International Operations Luxembourg S.A. (LU) 2007-12-26 EP claimed
WO-2006097460-A1 HYDROXAMATES AS HISTONE DEACETYLASE INHIBITORS AND PHARMACEUTICAL FORMULATIONS CONTAINING THEM MENARINI INTERNATIONAL OPERATIONS LUXEMBOURG S.A. (LU) 2006-09-21 WO claimed
EP-0740930-A1 BLOOD FLOW IMPROVER AND COSMETIC POLA CHEMICAL INDUSTRIES, INC. (JP) 1996-11-06 EP claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100069629-A1 PYRIMIDINE DERIVATIVES AS PI3K INHIBITOR AND USE THEREOF PIK3CA, AKT3, AKT1 CYP2A6 3158/4885CYP3A4 3027/4885ALDH1A1 2102/4885
US-20210145818-A1 COMPOSITIONS INFUSED WITH NICOTINE COMPOUNDS AND METHODS OF USE THEREOF CHRNA5, SLC18A3, CHRNA6 CYP2A6 1222/4885CYP3A4 1962/4885ALDH1A1 2986/4885
US-20080207694-A1 Hydroxamates as Histone Deacetylase Inhibitors and Pharmaceutical Formulations Containing Them HDAC1, HDAC8, HDAC9 CYP2A6 2796/4885CYP3A4 2599/4885ALDH1A1 1106/4885
US-20090258876-A1 NOVEL INDOL CARBOXYLIC ACID BISPYRIDYL CARBOXAMIDE DERIVATIVES, PHARMACEUTICALLY ACCEPTABLE SALT THEREOF, PREPARATION METHOD AND COMPOSITION CONTAINING THE SAME AS AN ACTIVE INGREDIENT HTR2C, HTR5A, HTR2A CYP2A6 1322/4885CYP3A4 806/4885ALDH1A1 1218/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.