SCHEMBL22556727

SCHEMBL22556727

COc1cccc(-c2cnc(CCl)o2)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
VCP P55072 1/20 0.52
FAAH O00519 1/20 0.48
HDAC1 Q13547 2/20 0.47
HDAC6 Q9UBN7 2/20 0.47
DYRK1A Q13627 1/20 0.46
CLK4 Q9HAZ1 1/20 0.46
FLT1 P17948 1/20 0.46
FLT4 P35916 1/20 0.46
KDR P35968 1/20 0.46
KDM4E B2RXH2 5/20 0.45
MAPT P10636 4/20 0.45
LMNA P02545 2/20 0.45
TDP1 Q9NUW8 1/20 0.45
ALDH1A1 P00352 5/20 0.44
HPGD P15428 5/20 0.44
SMN1; SMN2 Q16637 3/20 0.44
NPC1 O15118 3/20 0.44
MAPK1 P28482 2/20 0.44
RAB9A P51151 2/20 0.44
USP2 O75604 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29394070 1.00 VCP (0.52) VCPFAAHHDAC1HDAC6DYRK1A
SCHEMBL22556757 0.87 BRD4 (0.46) VCPKDM4EMAPTTDP1ALDH1A1
SCHEMBL22570681 0.82 PRMT1 (0.44) DYRK1ACYP3A4
SCHEMBL5639075 0.82 HDAC1 (0.53) FAAHHDAC1HDAC6KDM4EMAPT
SCHEMBL5472146 0.81 VCP (0.55) VCPFAAHHDAC1HDAC6DYRK1A
SCHEMBL22556766 0.80 NOTUM (0.40) VCPHDAC1HDAC6FLT1FLT4
SCHEMBL29393846 0.79 FFAR1 (0.52) VCPHDAC1HDAC6FLT1FLT4
SCHEMBL20600253 0.79 FFAR1 (0.52) VCPHDAC1HDAC6FLT1FLT4
SCHEMBL22556758 0.79 NOTUM (0.54) HDAC1HDAC6FLT1FLT4KDR
SCHEMBL2406093 0.79 VCP (0.56) VCPFAAHDYRK1ACLK4FLT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3956323-A1 OXAZOLE AND OXADIAZOLE DERIVATIVES USEFUL AS AGONISTS OF FREE FATTY ACID RECEPTOR 1 Gbiotech S.À.R.L. (CH) 2022-02-23 EP disclosed
WO-2020211956-A1 OXAZOLE AND OXADIAZOLE DERIVATIVES USEFUL AS AGONISTS OF FREE FATTY ACID RECEPTOR 1 GBIOTECH S.À.R.L. (CH) 2020-10-22 WO disclosed