SCHEMBL22561899

SCHEMBL22561899

C=C(Nc1ccc(C)c(-c2cnc(C3CCC3)c(C)c2)c1)c1cccc(SC)c1

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ADCY1 Q08828 1/20 0.37
ABL1 P00519 6/20 0.37
MAPK14 Q16539 2/20 0.34
MEN1 O00255 3/20 0.33
KMT2A Q03164 3/20 0.33
CYP1A2 P05177 2/20 0.33
CYP3A4 P08684 1/20 0.33
MAPT P10636 1/20 0.33
RHOA P61586 1/20 0.33
HCRTR1 O43613 1/20 0.33
HCRTR2 O43614 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
RAF1 P04049 4/20 0.33
BRAF P15056 3/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20009149 0.69 RAF1 (0.41) MAPTRAF1BRAF
SCHEMBL23677290 0.65 MEN1 (0.46) MEN1KMT2ACYP1A2CYP3A4MAPT
SCHEMBL25739849 0.64 SMN1; SMN2 (0.62) MEN1KMT2ACYP1A2CYP3A4MAPT
SCHEMBL20009394 0.60 BRAF (0.70) MAPK14RAF1BRAF
SCHEMBL14305900 0.60 LDLR (0.38) MAPK14
SCHEMBL26949118 0.57 ABL1 (0.46) ABL1MEN1KMT2A
SCHEMBL22490321 0.57 MAPK14 (0.59) ABL1MAPK14CYP2C9RAF1
SCHEMBL1990577 0.56
SCHEMBL1990574 0.56
SCHEMBL29536688 0.56

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3191467-B1 COMPOUNDS AND COMPOSITIONS AS KINASE INHIBITORS NOVARTIS AG (CH) 2020-10-21 EP disclosed