SCHEMBL22561941

SCHEMBL22561941

CNc1ccc(C)c(-c2cnc(N3CCNCC3)c(C#N)c2)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RET P07949 8/20 0.48
CNR2 P34972 1/20 0.44
TAAR1 Q96RJ0 1/20 0.44
CYP1A2 P05177 3/20 0.41
CYP3A4 P08684 3/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
TSHR P16473 2/20 0.41
CYP2D6 P10635 1/20 0.41
RECQL P46063 1/20 0.41
CDK9 P50750 4/20 0.41
CDC7 O00311 1/20 0.41
PIM1 P11309 1/20 0.41
CCNT1 O60563 3/20 0.40
CCNA2 P20248 3/20 0.40
CDK2 P24941 3/20 0.40
CDK1 P06493 2/20 0.40
CCNB1 P14635 2/20 0.40
CDK7 P50613 2/20 0.40
CCNH P51946 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22561868 0.81 RAF1 (0.51)
SCHEMBL19328136 0.78 RAF1 (0.57)
SCHEMBL19328040 0.77 RAF1 (0.59)
SCHEMBL19328082 0.77 RAF1 (0.65)
SCHEMBL19327905 0.77 RAF1 (0.57)
SCHEMBL19328074 0.77 RAF1 (0.55)
SCHEMBL19327912 0.77 RAF1 (0.57)
SCHEMBL19327942 0.77 BRAF (0.56)
SCHEMBL19327962 0.77 RAF1 (0.58)
SCHEMBL19327935 0.77 RAF1 (0.56)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3191467-B1 COMPOUNDS AND COMPOSITIONS AS KINASE INHIBITORS NOVARTIS AG (CH) 2020-10-21 EP disclosed