SCHEMBL22604349

SCHEMBL22604349

Cc1cn(-c2cccc(C(C)(C)C)c2)cn1

nearest known ligand 0.52

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP2E1 P05181 1/20 0.51
CYP2A6 P11509 1/20 0.51
NR2E1 Q9Y466 9/20 0.49
MAOA P21397 1/20 0.43
MAOB P27338 1/20 0.43
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP19A1 P11511 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
NOTUM Q6P988 1/20 0.40
MAPK13 O15264 1/20 0.40
OPRM1 P35372 1/20 0.40
OPRD1 P41143 1/20 0.40
OPRK1 P41145 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12907213 0.86 NR2E1 (0.45) CYP2E1CYP2A6NR2E1CYP1A2CYP3A4
SCHEMBL15381990 0.86 NR2E1 (0.62) CYP2E1CYP2A6NR2E1CYP1A2NOTUM
SCHEMBL12372948 0.83 NR2E1 (0.58) CYP2E1CYP2A6NR2E1MAOAMAOB
SCHEMBL18120009 0.80 NPC1 (0.54) MAOAMAOBNOTUMOPRM1OPRD1
SCHEMBL270618 0.80 CYP1A2 (0.53) CYP2E1CYP2A6NR2E1MAOAMAOB
SCHEMBL4426922 0.79 NOTUM (0.43) NOTUMOPRM1OPRD1OPRK1
SCHEMBL15315567 0.79 NR2E1 (0.54) CYP2E1CYP2A6NR2E1CYP1A2CYP3A4
SCHEMBL23510668 0.78 MAP3K5 (0.45)
Phosphoric Acid SCHEMBL28774218 0.78 NR2E1 (0.55) NR2E1CYP1A2
SCHEMBL21849237 0.78 OPRD1 (0.44) CYP1A2CYP2C9NOTUMOPRM1OPRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020216071-A1 DIMERIC OR POLYMERIC FORM OF MUTANT IDH INHIBITOR 上海仕谱生物科技有限公司 2020-10-29 WO disclosed