SCHEMBL22607649

SCHEMBL22607649

NC(=O)CCN1CCOC1=O

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.41
NAAA Q02083 7/20 0.39
CNR1 P21554 1/20 0.37
CNR2 P34972 1/20 0.37
ALDH1A1 P00352 1/20 0.37
LMNA P02545 1/20 0.37
POLB P06746 1/20 0.37
MAPT P10636 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
KMT2A Q03164 1/20 0.37
PIK3CD O00329 1/20 0.36
CYP11B2 P19099 1/20 0.35
TSHR P16473 1/20 0.34
MAPK1 P28482 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
FAAH O00519 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17662299 0.83 KDM4E (0.45) KDM4EL3MBTL1NAAACNR1CNR2
SCHEMBL4787017 0.81 TSHR (0.48) KDM4ENAAAPIK3CDTSHRMAPK1
SCHEMBL9310220 0.79 KDM4E (0.38) KDM4ENAAACNR1CNR2ALDH1A1
SCHEMBL20329218 0.77 KDM4E (0.41) KDM4ENAAACNR1CNR2ALDH1A1
SCHEMBL9310675 0.77 KMT2A (0.45) KDM4ENAAACNR1CNR2ALDH1A1
SCHEMBL20105 0.76
SCHEMBL510011 0.76
SCHEMBL6378864 0.76 ALDH1A1 (0.44) KDM4EL3MBTL1NAAAALDH1A1LMNA
Hydrochloric Acid SCHEMBL18050151 0.75 KDM4E (0.47) KDM4ENAAACNR1CNR2ALDH1A1
SCHEMBL1712876 0.74

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3013832-B1 PYRAZOLE COMPOUNDS AS MODULATORS OF FSHR AND USES THEREOF MERCK PATENT GMBH (DE) 2020-11-04 EP disclosed