SCHEMBL22609986

SCHEMBL22609986

COC1(OC)CC(C#N)C1

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28066082 0.78
SCHEMBL16636031 0.74
SCHEMBL25309239 0.70
SCHEMBL25309241 0.70
SCHEMBL9143364 0.69
SCHEMBL26116030 0.69
SCHEMBL8738683 0.67
SCHEMBL25299741 0.66
SCHEMBL17621627 0.65
SCHEMBL13455883 0.65

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 18 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4499634-A1 SULFONAMIDO DERIVATIVES AS CYCLIN-DEPENDENT KINASE 2 INHIBITORS Nikang Therapeutics, Inc. (US) 2025-02-05 EP disclosed
CN-119053595-A Sulfonylamino derivatives as cyclin dependent kinase 2 inhibitors 尼坎治疗公司 2024-11-29 CN disclosed
WO-2024064745-A1 SYNTHESIS OF RELDESEMTIV CYTOKINETICS, INCORPORATED (US) 2024-03-28 WO disclosed
WO-2024017178-A1 SUBSTITUTED HYDANTOIN COMPOUNDS, PHARMACEUTICAL COMPOSITIONS, AND THERAPEUTIC APPLICATIONS AVITAR BIOSCIENCES, INC. (CN) 2024-01-25 WO disclosed
CN-112236415-B Process for the preparation of aminopyrimidines and intermediates therefor 赛特凯恩蒂克公司 2023-11-14 CN disclosed
WO-2023192801-A1 SULFONAMIDO DERIVATIVES AS CYCLIN-DEPENDENT KINASE 2 INHIBITORS NIKANG THERAPEUTICS, INC. (US) 2023-10-05 WO disclosed
US-20230303509-A1 SULFONAMIDO DERIVATIVES AS CYCLIN-DEPENDENT KINASE 2 INHIBITORS NIKANG THERAPEUTICS, INC. 2023-09-28 US disclosed
US-20230303509-A1 SULFONAMIDO DERIVATIVES AS CYCLIN-DEPENDENT KINASE 2 INHIBITORS NIKANG THERAPEUTICS, INC. 2023-09-28 US disclosed
WO-2023151642-A1 HETEROCYCLIC COMPOUNDS, COMPOSITIONS THEREOF, AND METHODS OF TREATMENT THEREWITH BEIGENE , LTD. (KY) 2023-08-17 WO disclosed
WO-2023151636-A1 HETEROCYCLIC COMPOUNDS, COMPOSITIONS THEREOF, AND METHODS OF TREATMENT THEREWITH BEIGENE , LTD. (KY) 2023-08-17 WO disclosed
WO-2023151641-A1 HETEROCYCLIC COMPOUNDS, COMPOSITIONS THEREOF, AND METHODS OF TREATMENT THEREWITH BEIGENE , LTD. (KY) 2023-08-17 WO disclosed
WO-2023151640-A1 HETEROCYCLIC COMPOUNDS, COMPOSITIONS THEREOF, AND METHODS OF TREATMENT THEREWITH BEIGENE , LTD. (KY) 2023-08-17 WO disclosed
US-11142516-B2 Process for the preparation of an amino-pyrimidine and intermediates thereof CYTOKINETICS, INC. (US) 2021-10-12 US disclosed
US-11142516-B2 Process for the preparation of an amino-pyrimidine and intermediates thereof CYTOKINETICS, INC. (US) 2021-10-12 US disclosed
US-20210061786-A1 PROCESS FOR THE PREPARATION OF AN AMINO-PYRIMIDINE AND INTERMEDIATES THEREOF CYTOKINETICS, INC. (US) 2021-03-04 US disclosed
US-20210061786-A1 PROCESS FOR THE PREPARATION OF AN AMINO-PYRIMIDINE AND INTERMEDIATES THEREOF CYTOKINETICS, INC. (US) 2021-03-04 US disclosed
CN-112236415-A Process for preparing aminopyrimidines and intermediates thereof 赛特凯恩蒂克公司 2021-01-15 CN disclosed
EP-3732166-A1 PROCESS FOR THE PREPARATION OF AN AMINO-PYRIMIDINE AND INTERMEDIATES THEREOF Cytokinetics, Incorporated (US) 2020-11-04 EP disclosed