SCHEMBL22620109

SCHEMBL22620109

CC(C)(C)OC(=O)N1CCC[C@@H](Nc2c(Br)cnc3c2ccn3COCC[Si](C)(C)C)C1

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HDAC4 P56524 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
BCHE P06276 2/20 0.39
HTR6 P50406 2/20 0.39
USP30 Q70CQ3 4/20 0.38
PIK3CD O00329 1/20 0.37
GABRA5 P31644 1/20 0.37
FPR3 P25089 1/20 0.37
FPR2 P25090 1/20 0.37
BTK Q06187 2/20 0.36
ANO1 Q5XXA6 1/20 0.36
IGF1R P08069 1/20 0.36
BRD4 O60885 1/20 0.35
JAK2 O60674 1/20 0.35
JAK1 P23458 1/20 0.35
PARP1 P09874 1/20 0.35
TRPV3 Q8NET8 1/20 0.35
PBK Q96KB5 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29855767 1.00 HDAC4 (0.40) HDAC4HDAC6BCHEHTR6USP30
SCHEMBL22613075 0.90 BCHE (0.40) HDAC4HDAC6BCHEHTR6USP30
SCHEMBL22613074 0.90 BCHE (0.40) HDAC4HDAC6BCHEHTR6USP30
SCHEMBL10099184 0.90 HTR6 (0.40) HDAC4HDAC6BCHEHTR6USP30
SCHEMBL22613184 0.90 JAK3 (0.34) JAK2JAK1
SCHEMBL22613183 0.90 JAK3 (0.34) JAK2JAK1
SCHEMBL10099173 0.89 JAK3 (0.45) HDAC4HDAC6BCHEHTR6USP30
SCHEMBL22620168 0.88 JAK3 (0.49) JAK1
SCHEMBL22620101 0.88 JAK3 (0.49) JAK1
SCHEMBL22620117 0.87 JAK2 (0.46) HDAC4HDAC6BCHEHTR6USP30

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020223728-A1 SUBSTITUTED PYRROLOPYRIDINES AS JAK INHIBITORS ACLARIS THERAPEUTICS, INC. (US) 2020-11-05 WO disclosed