SCHEMBL22620199

SCHEMBL22620199

CC1CC(NC(=O)OC(C)(C)C)CN(C)C1

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CTSK P43235 2/20 0.47
BTK Q06187 1/20 0.47
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
HSD11B1 P28845 4/20 0.42
CYP2C9 P11712 1/20 0.42
EIF2AK4 Q9P2K8 1/20 0.40
AURKA O14965 1/20 0.40
PDPK1 O15530 1/20 0.40
AURKB Q96GD4 1/20 0.40
KMT2A Q03164 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
GAA P10253 1/20 0.39
KDM1A O60341 1/20 0.39
MAOB P27338 1/20 0.39
EPHX2 P34913 1/20 0.38
NFKB1 P19838 1/20 0.38
NFKB2 Q00653 1/20 0.38
RELA Q04206 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12814322 0.87 CTSK (0.54) CTSKBTKCA1CA2HSD11B1
SCHEMBL24087331 0.84 CTSK (0.47) CTSKBTKCA1CA2HSD11B1
SCHEMBL24076246 0.84 CTSK (0.47) CTSKBTKCA1CA2HSD11B1
SCHEMBL30054708 0.83 CTSK (0.46) CTSKBTKCA1CA2HSD11B1
SCHEMBL25085897 0.83 CTSK (0.46) CTSKBTKCA1CA2HSD11B1
SCHEMBL17859548 0.83 CTSK (0.46) CTSKBTKCA1CA2HSD11B1
SCHEMBL17859549 0.83 CTSK (0.46) CTSKBTKCA1CA2HSD11B1
SCHEMBL16665756 0.83 CTSK (0.46) CTSKBTKCA1CA2HSD11B1
SCHEMBL24087333 0.82 CTSK (0.45) CTSKBTKCA1CA2HSD11B1
SCHEMBL20498700 0.82 BTK (0.48) CTSKBTKCA1CA2HSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020223728-A1 SUBSTITUTED PYRROLOPYRIDINES AS JAK INHIBITORS ACLARIS THERAPEUTICS, INC. (US) 2020-11-05 WO disclosed