SCHEMBL22622754

SCHEMBL22622754

Cc1cc(-c2ccc(C#Cc3ccc(OC(F)(F)F)cc3)cc2)cc(F)c1N=C=S

nearest known ligand 0.36

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ACACB O00763 1/20 0.34
AURKA O14965 1/20 0.34
TPX2 Q9ULW0 1/20 0.34
PPARD Q03181 2/20 0.33
SCN5A Q14524 2/20 0.33
PTGER4 P35408 1/20 0.33
KIF11 P52732 1/20 0.33
FFAR4 Q5NUL3 2/20 0.33
FFAR1 O14842 1/20 0.33
AKR1C2 P52895 1/20 0.32
AKR1C1 Q04828 1/20 0.32
DHODH Q02127 1/20 0.32
KDM4E B2RXH2 1/20 0.32
GAA P10253 1/20 0.32
MAPT P10636 1/20 0.32
MAPK1 P28482 1/20 0.32
PRMT6 Q96LA8 1/20 0.32
GRIN2B Q13224 1/20 0.32
NAAA Q02083 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22622797 0.93 ACACB (0.34) ACACBAURKATPX2PPARDSCN5A
SCHEMBL22622985 0.91 AURKA (0.37) ACACBAURKATPX2SCN5AKIF11
SCHEMBL22622867 0.89 ACACB (0.33) ACACBAURKATPX2SCN5AFFAR4
SCHEMBL22622826 0.86 ACACB (0.35) ACACBAURKATPX2PPARDSCN5A
SCHEMBL22622815 0.86 ACACB (0.35) ACACBAURKATPX2SCN5APTGER4
SCHEMBL22622976 0.85 DHODH (0.31) SCN5APTGER4KIF11DHODHNAAA
SCHEMBL22622974 0.85 AURKA (0.31) AURKATPX2SCN5APTGER4KIF11
SCHEMBL24390836 0.85 KCNH2 (0.32) NAAA
SCHEMBL25056671 0.85 AURKA (0.41) AURKATPX2SCN5AKIF11AKR1C2
SCHEMBL22622688 0.83 ACACB (0.33) ACACBAURKATPX2SCN5AFFAR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022090098-A1 AROMATIC ISOTHIOCYANATES MERCK PATENT GMBH (DE) 2022-05-05 WO disclosed
US-20200347301-A1 Isothiocyanato-tolanes MERCK PATENT GMBH (DE) 2020-11-05 US disclosed
EP-3733816-A1 ISOTHIOCYANATO-TOLANES Merck Patent GmbH (DE) 2020-11-04 EP disclosed