SCHEMBL22622985

SCHEMBL22622985

Fc1cc(-c2ccc(C#Cc3ccc(OC(F)(F)F)cc3)cc2)cc(F)c1N=C=S

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AURKA O14965 1/20 0.37
TPX2 Q9ULW0 1/20 0.37
AKR1C2 P52895 1/20 0.35
AKR1C1 Q04828 1/20 0.35
ACACB O00763 1/20 0.35
DHODH Q02127 1/20 0.34
SCN5A Q14524 6/20 0.34
KIF11 P52732 2/20 0.34
EPM2A O95278 1/20 0.33
PTPRC P08575 1/20 0.33
PTPN2 P17706 1/20 0.33
PTPN1 P18031 1/20 0.33
PTPRG P23470 1/20 0.33
ACP1 P24666 1/20 0.33
PTPN6 P29350 1/20 0.33
PTPN7 P35236 1/20 0.33
PTPN9 P43378 1/20 0.33
DUSP3 P51452 1/20 0.33
PTPN11 Q06124 1/20 0.33
PTPN13 Q12923 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22622815 0.95 ACACB (0.35) AURKATPX2AKR1C2AKR1C1ACACB
SCHEMBL25056671 0.93 AURKA (0.41) AURKATPX2AKR1C2AKR1C1DHODH
SCHEMBL22622754 0.91 ACACB (0.34) AURKATPX2AKR1C2AKR1C1ACACB
SCHEMBL22622688 0.91 ACACB (0.33) AURKATPX2AKR1C2AKR1C1ACACB
SCHEMBL26383670 0.90 ACACB (0.37) ACACBKIF11EPM2APTPRCPTPN2
SCHEMBL22622831 0.90 ACACB (0.37) ACACBKIF11EPM2APTPRCPTPN2
SCHEMBL22622867 0.87 ACACB (0.33) AURKATPX2ACACBDHODHSCN5A
SCHEMBL22622826 0.87 ACACB (0.35) AURKATPX2ACACBSCN5ATRPA1
SCHEMBL22622797 0.86 ACACB (0.34) AURKATPX2ACACBSCN5AKIF11
SCHEMBL22622802 0.86 SCN5A (0.33) AURKATPX2DHODHSCN5AKIF11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230313043-A1 OPTICAL COMPONENT MERCK PATENT GMBH (DE) 2023-10-05 US disclosed
US-20200347301-A1 Isothiocyanato-tolanes MERCK PATENT GMBH (DE) 2020-11-05 US disclosed
EP-3733816-A1 ISOTHIOCYANATO-TOLANES Merck Patent GmbH (DE) 2020-11-04 EP disclosed