SCHEMBL22637851

SCHEMBL22637851

COc1cccc(-c2noc(C(C)NC(=O)O)n2)c1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S1PR3 Q99500 1/20 0.60
ACACB O00763 5/20 0.57
PPARD Q03181 4/20 0.57
PPARA Q07869 4/20 0.57
RECQL P46063 1/20 0.54
NPC1 O15118 3/20 0.53
RAB9A P51151 3/20 0.53
TDP1 Q9NUW8 2/20 0.53
TP53 P04637 2/20 0.53
SMN1; SMN2 Q16637 2/20 0.53
NFKB1 P19838 1/20 0.53
NFKB2 Q00653 1/20 0.53
RELA Q04206 1/20 0.53
IDH1 O75874 1/20 0.51
TUBB4A P04350 2/20 0.51
TUBB P07437 2/20 0.51
TUBA3C P0DPH7 2/20 0.51
TUBA1B P68363 2/20 0.51
TUBA4A P68366 2/20 0.51
TUBB4B P68371 2/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22637849 1.00 S1PR3 (0.60) S1PR3ACACBPPARDPPARARECQL
SCHEMBL22649322 0.86 PPARD (0.53) S1PR3ACACBPPARDPPARARECQL
SCHEMBL29463559 0.86 PPARD (0.53) S1PR3ACACBPPARDPPARARECQL
SCHEMBL22637723 0.85 KCNT1 (0.64) ACACBPPARDPPARARAB9ATDP1
SCHEMBL22637840 0.85 KCNT1 (0.64) ACACBPPARDPPARARAB9ATDP1
SCHEMBL22637724 0.85 KCNT1 (0.64) ACACBPPARDPPARARAB9ATDP1
SCHEMBL22637923 0.84 TDP1 (0.56) ACACBPPARDPPARATDP1TP53
SCHEMBL22637891 0.83 KCNT1 (0.64) ACACBPPARDPPARATDP1TP53
SCHEMBL22637893 0.83 KCNT1 (0.64) ACACBPPARDPPARATDP1TP53
SCHEMBL22637761 0.83 TDP1 (0.55) ACACBPPARDPPARANPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3962481-A1 KCNT1 INHIBITORS AND METHODS OF USE Praxis Precision Medicines, Inc. (US) 2022-03-09 EP disclosed
WO-2020227101-A1 KCNT1 INHIBITORS AND METHODS OF USE PRAXIS PRECISION MEDICINES, INC. (US) 2020-11-12 WO disclosed