SCHEMBL22650363

SCHEMBL22650363

CCN1CCN(c2ccc(Nc3nccc(-c4ccn5ncc(C(C)C)c5c4)n3)nc2)C(=O)C1

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
BTK Q06187 8/20 0.44
CDK4 P11802 11/20 0.42
CDK1 P06493 9/20 0.42
CCND1 P24385 9/20 0.42
CCNB1 P14635 7/20 0.42
CDK6 Q00534 5/20 0.42
DYRK2 Q92630 1/20 0.41
CCND3 P30281 3/20 0.39
CCNA2 P20248 5/20 0.38
CDK2 P24941 5/20 0.38
CCNA1 P78396 4/20 0.38
CCNT1 O60563 1/20 0.38
CDK7 P50613 1/20 0.38
CDK9 P50750 1/20 0.38
CCNH P51946 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22650862 0.92 CDK4 (0.46) BTKCDK4CDK1CCND1CCNB1
SCHEMBL22650602 0.87 CDK6 (0.46) CDK4CDK1CCND1CCNB1CDK6
SCHEMBL22650361 0.85 BTK (0.40) BTKCDK4CDK1CCND1CCNB1
SCHEMBL22650569 0.85 CDK4 (0.43) BTKCDK4CDK1CCND1CCNB1
SCHEMBL29491175 0.85 CDK4 (0.49) CDK4CDK1CCND1CCNB1CDK6
SCHEMBL22650568 0.85 CDK4 (0.49) CDK4CDK1CCND1CCNB1CDK6
SCHEMBL22650846 0.85 CDK4 (0.42) CDK4CDK1CCND1CCNB1CDK6
SCHEMBL22650924 0.84 CDK4 (0.48) CDK4CDK1CCND1CCNB1CDK6
SCHEMBL22650472 0.84 CDK4 (0.45) BTKCDK4CDK1CCND1CCNB1
SCHEMBL22650755 0.84 CDK4 (0.42) CDK4CDK1CCND1CCNB1CDK6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020224568-A1 CDK INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2020-11-12 WO disclosed