SCHEMBL22650846

SCHEMBL22650846

CC(C)c1cnn2ccc(-c3ccnc(Nc4ccc(N5CCOCC5=O)cn4)n3)cc12

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 11/20 0.42
CDK6 Q00534 9/20 0.42
CCND1 P24385 7/20 0.42
CDK1 P06493 6/20 0.42
CCNB1 P14635 5/20 0.42
TYK2 P29597 2/20 0.42
CCNA2 P20248 5/20 0.41
CCND3 P30281 5/20 0.41
CDK2 P24941 4/20 0.41
JAK2 O60674 6/20 0.40
JAK3 P52333 3/20 0.40
JAK1 P23458 1/20 0.40
CCNA1 P78396 3/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22650922 0.87 F10 (0.38) TYK2JAK2JAK3JAK1
SCHEMBL22650591 0.87 CDK6 (0.48) CDK4CDK6CCND1CDK1CCNB1
SCHEMBL22650568 0.86 CDK4 (0.49) CDK4CDK6CCND1CDK1CCNB1
SCHEMBL29491175 0.86 CDK4 (0.49) CDK4CDK6CCND1CDK1CCNB1
SCHEMBL22650924 0.86 CDK4 (0.48) CDK4CDK6CCND1CDK1CCNB1
SCHEMBL22650755 0.85 CDK4 (0.42) CDK4CDK6CCND1CDK1CCNB1
SCHEMBL22650361 0.85 BTK (0.40) CDK4CDK6CCND1CDK1CCNB1
SCHEMBL22650453 0.85 CDK4 (0.42) CDK4CDK6CCND1CDK1CCNB1
SCHEMBL22650485 0.85 CDK4 (0.47) CDK4CDK6CCND1CDK1CCNB1
SCHEMBL22650363 0.85 BTK (0.44) CDK4CDK6CCND1CDK1CCNB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020224568-A1 CDK INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2020-11-12 WO disclosed