SCHEMBL22650421

SCHEMBL22650421

CC(C)c1cnn2ccc(-c3ccnc(Nc4ccc(N5CCC(N(C)C)CC5=O)cc4)n3)cc12

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 8/20 0.38
JAK3 P52333 6/20 0.38
IKBKB O14920 1/20 0.37
CHUK O15111 1/20 0.37
IKBKG Q9Y6K9 1/20 0.37
CDK4 P11802 3/20 0.37
CCND1 P24385 3/20 0.37
CCNA2 P20248 3/20 0.37
CDK2 P24941 3/20 0.37
CCNA1 P78396 3/20 0.37
GSK3B P49841 1/20 0.37
JAK1 P23458 1/20 0.36
EGFR P00533 3/20 0.36
CDK1 P06493 1/20 0.36
CCNB1 P14635 1/20 0.36
ABL1 P00519 1/20 0.35
PDGFRB P09619 1/20 0.35
BCR P11274 1/20 0.35
SRC P12931 1/20 0.35
PDGFRA P16234 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22650901 0.91 CDK4 (0.45) CDK4CCND1CCNA2CDK2CCNA1
SCHEMBL22650823 0.91 CDK4 (0.45) CDK4CCND1CCNA2CDK2CCNA1
SCHEMBL22650597 0.89 EGFR (0.37) JAK2JAK3CDK4CCND1CCNA2
SCHEMBL22650847 0.88 JAK2 (0.39) JAK2JAK3CDK4CCND1CCNA2
SCHEMBL22650423 0.86 JAK2 (0.37) JAK2JAK3IKBKBCHUKIKBKG
SCHEMBL22650419 0.85 JAK2 (0.38) JAK2JAK3CDK4CCND1JAK1
SCHEMBL22650434 0.85 JAK2 (0.36) JAK2JAK3CDK4CCND1CDK2
SCHEMBL22650417 0.84 CDK4 (0.40) CDK4CCND1CCNA2CDK2CCNA1
SCHEMBL22650526 0.83 MAP4K1 (0.44) JAK2JAK3IKBKBCHUKCDK4
SCHEMBL22650851 0.83 IKBKB (0.56) IKBKBCHUKIKBKGCDK2CDK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020224568-A1 CDK INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2020-11-12 WO disclosed