SCHEMBL22650423

SCHEMBL22650423

Cc1nn2ccc(-c3ccnc(Nc4ccc(N5CCC(N(C)C)CC5=O)cc4)n3)cc2c1C(C)C

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 10/20 0.37
JAK3 P52333 5/20 0.37
MAPK8 P45983 1/20 0.37
MAPK10 P53779 1/20 0.37
IKBKB O14920 1/20 0.37
CHUK O15111 1/20 0.37
IKBKG Q9Y6K9 1/20 0.37
CDK4 P11802 2/20 0.36
CCND1 P24385 2/20 0.36
CDK1 P06493 1/20 0.36
CCNB1 P14635 1/20 0.36
ABL1 P00519 2/20 0.35
PDGFRB P09619 2/20 0.35
KIT P10721 2/20 0.35
EGFR P00533 2/20 0.35
CCNA2 P20248 1/20 0.35
CDK2 P24941 1/20 0.35
GSK3B P49841 1/20 0.35
CCNA1 P78396 1/20 0.35
BRD4 O60885 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22650421 0.86 JAK2 (0.38) JAK2JAK3IKBKBCHUKIKBKG
SCHEMBL22650604 0.85 JAK2 (0.37) JAK2JAK3MAPK8MAPK10CDK4
SCHEMBL22650701 0.82 JAK2 (0.38) JAK2JAK3MAPK8MAPK10CDK4
SCHEMBL22650716 0.82 JAK2 (0.38) JAK2JAK3MAPK8MAPK10CDK4
SCHEMBL22650901 0.77 CDK4 (0.45) CDK4CCND1CDK1CCNB1CCNA2
SCHEMBL22650823 0.77 CDK4 (0.45) CDK4CCND1CDK1CCNB1CCNA2
SCHEMBL22650597 0.76 EGFR (0.37) JAK2JAK3MAPK8CDK4CCND1
SCHEMBL22650781 0.74 IKBKB (0.39) JAK2JAK3IKBKBCHUKIKBKG
SCHEMBL22650930 0.74 CDK4 (0.50) CDK4CCND1CDK1CCNB1CCNA2
SCHEMBL22650847 0.74 JAK2 (0.39) JAK2JAK3CDK4CCND1CDK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020224568-A1 CDK INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2020-11-12 WO disclosed