SCHEMBL22650463

SCHEMBL22650463

COc1nc(-c2ccnc(Nc3ccc(N4CC5CC4CN5)cn3)n2)cc2c1ncn2C(C)C

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 8/20 0.44
CCND1 P24385 7/20 0.44
CDK6 Q00534 2/20 0.44
CHRNB2 P17787 10/20 0.43
CHRNA4 P43681 10/20 0.43
CDK1 P06493 6/20 0.43
CCNT1 O60563 1/20 0.38
CDK9 P50750 1/20 0.38
CCNB1 P14635 5/20 0.36
CCNA2 P20248 4/20 0.36
CDK2 P24941 4/20 0.36
CCNA1 P78396 4/20 0.36
CHRNB4 P30926 1/20 0.35
CHRNA3 P32297 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22650577 0.90 CDK4 (0.48) CDK4CCND1CDK6CHRNB2CHRNA4
SCHEMBL22650510 0.85 CDK4 (0.37) CDK4CCND1CDK6CDK1CCNT1
SCHEMBL22650511 0.85 CCND1 (0.35) CDK4CCND1CDK6CDK1CCNT1
SCHEMBL22650859 0.80 CDK4 (0.51) CDK4CCND1CDK6CDK1CCNT1
SCHEMBL22650615 0.79 CDK4 (0.46) CDK4CCND1CDK6CDK1CCNT1
SCHEMBL22650546 0.79 CDK4 (0.42) CDK4CCND1CDK6CDK1CCNT1
SCHEMBL22650958 0.77 CDK4 (0.42) CDK4CCND1CDK6CDK1CCNT1
SCHEMBL22650548 0.77 CDK4 (0.41) CDK4CCND1CDK6CDK1CCNT1
SCHEMBL22650514 0.76 CDK4 (0.38) CDK4CCND1CDK6CDK1CCNT1
SCHEMBL22650513 0.75 CDK4 (0.36) CDK4CCND1CDK6CDK1CCNT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020224568-A1 CDK INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2020-11-12 WO disclosed