SCHEMBL22650577

SCHEMBL22650577

CC(C)n1cnc2c(F)nc(-c3ccnc(Nc4ccc(N5CC6CC5CN6)cn4)n3)cc21

nearest known ligand 0.48

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 12/20 0.48
CCND1 P24385 7/20 0.48
CDK6 Q00534 3/20 0.48
CDK1 P06493 7/20 0.43
CHRNB2 P17787 6/20 0.42
CHRNA4 P43681 6/20 0.42
CCNT1 O60563 1/20 0.38
CDK9 P50750 1/20 0.38
CCNB1 P14635 5/20 0.37
CCNA2 P20248 5/20 0.37
CDK2 P24941 4/20 0.37
CCNA1 P78396 4/20 0.37
CCND3 P30281 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22650463 0.90 CDK4 (0.44) CDK4CCND1CDK6CDK1CHRNB2
SCHEMBL22650628 0.80 CDK4 (0.58) CDK4CCND1CDK6CDK1CCNT1
SCHEMBL22650616 0.80 CDK6 (0.46) CDK4CCND1CDK6CDK1CCNT1
SCHEMBL22650607 0.80 CDK4 (0.46) CDK4CCND1CDK6CDK1CCNT1
SCHEMBL22650622 0.80 CDK4 (0.52) CDK4CCND1CDK6CDK1CCNT1
SCHEMBL22650778 0.78 CDK4 (0.42) CDK4CCND1CDK6CDK1CCNT1
SCHEMBL22650722 0.78 CDK4 (0.44) CDK4CCND1CDK6CDK1CCNT1
SCHEMBL22650579 0.77 CDK4 (0.48) CDK4CCND1CDK6CDK1CCNT1
SCHEMBL22650723 0.76 CDK4 (0.48) CDK4CCND1CDK6CDK1CCNT1
SCHEMBL22650875 0.75 TYK2 (0.44) CDK4CCND1CDK6CDK1CCNT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020224568-A1 CDK INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2020-11-12 WO disclosed