SCHEMBL22650585

SCHEMBL22650585

Cc1ccc2c(c1C)OCc1c-2ccc(C)c1I

nearest known ligand 0.51

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 2/20 0.51
ESR2 Q92731 2/20 0.51
PGR P06401 4/20 0.33
TDP2 O95551 1/20 0.33
NSD2 O96028 1/20 0.33
HSP90AA1 P07900 1/20 0.33
PAX8 Q06710 1/20 0.33
KCNJ1 P48048 1/20 0.32
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
HPGD P15428 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23849173 0.89 ESR1 (0.46) ESR1ESR2PGRKCNJ1
SCHEMBL21451571 0.86 ESR1 (0.51) ESR1ESR2PGRKCNJ1
SCHEMBL803200 0.85 ESR1 (0.62) ESR1ESR2PGRTDP2NSD2
SCHEMBL23289004 0.82 ESR1 (0.42) ESR1ESR2KCNJ1
SCHEMBL22644204 0.82 ESR1 (0.43) ESR1ESR2KCNJ1
SCHEMBL802785 0.76 ESR1 (0.51) ESR1ESR2PGRTDP2NSD2
SCHEMBL803047 0.74 ESR1 (0.50) ESR1ESR2PGRTDP2NSD2
SCHEMBL14883992 0.71 PSMB5 (0.52) ESR1ESR2TDP2NSD2HSP90AA1
SCHEMBL23284915 0.70 ESR1 (0.44) ESR1ESR2TDP2NSD2HSP90AA1
SCHEMBL14883956 0.68 PSMB5 (0.49) ESR1ESR2TDP2NSD2HSP90AA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3481916-B1 ELECTRONIC SWITCH MERCK PATENT GMBH (DE) 2021-11-03 EP disclosed
WO-2020225398-A1 AROMATIC COMPOUNDS MERCK PATENT GMBH (DE) 2020-11-12 WO disclosed