SCHEMBL22650614

SCHEMBL22650614

CCN1CCN(Cc2ccc(Nc3ncc(F)c(-c4cc5c(nc(C)n5C(C)C)c(OC)n4)n3)nc2)CC1

nearest known ligand 0.75

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK6 Q00534 15/20 0.75
CDK4 P11802 11/20 0.75
CCND1 P24385 9/20 0.75
CCND3 P30281 7/20 0.75
CDK1 P06493 7/20 0.75
CCNA2 P20248 5/20 0.75
CDK2 P24941 5/20 0.75
CCNE2 O96020 4/20 0.75
PIM1 P11309 2/20 0.75
DYRK2 Q92630 2/20 0.75
CIT O14578 1/20 0.75
GAK O14976 1/20 0.75
DYRK3 O43781 1/20 0.75
CCNT1 O60563 1/20 0.75
STK16 O75716 1/20 0.75
CCNK O75909 1/20 0.75
STK10 O94804 1/20 0.75
PRKD3 O94806 1/20 0.75
ABCB11 O95342 1/20 0.75
MAP4K4 O95819 1/20 0.75

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22650956 0.87 CDK6 (0.59) CDK6CDK4CCND1CCND3CDK1
SCHEMBL22650635 0.87 CDK6 (0.57) CDK6CDK4CCND1CCND3CDK1
Abemaciclib SCHEMBL29356350 0.86 CDK4 (1.00) CDK6CDK4CCND1CCND3CDK1
Abemaciclib SCHEMBL2487229 0.86 CDK4 (1.00) CDK6CDK4CCND1CCND3CDK1
Abemaciclib SCHEMBL29423472 0.86 CDK4 (1.00) CDK6CDK4CCND1CCND3CDK1
Abemaciclib SCHEMBL29591527 0.86 CDK4 (1.00) CDK6CDK4CCND1CCND3CDK1
SCHEMBL19057207 0.85 CDK6 (0.90) CDK6CDK4CCND1CCND3CDK1
SCHEMBL22650452 0.85 CDK4 (0.54) CDK6CDK4CCND1CCND3CDK1
SCHEMBL26840566 0.84 CDK6 (0.78) CDK6CDK4CCND1CCND3CDK1
SCHEMBL24021429 0.84 CDK4 (0.95) CDK6CDK4CCND1CCND3CDK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020224568-A1 CDK INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2020-11-12 WO disclosed