SCHEMBL22650635

SCHEMBL22650635

COc1nc(-c2nc(Nc3ccc(CN4CCN5CCCC5C4)cn3)ncc2F)cc2c1nc(C)n2C(C)C

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK6 Q00534 17/20 0.57
CDK4 P11802 14/20 0.57
CCND1 P24385 7/20 0.57
CDK1 P06493 6/20 0.57
CCND3 P30281 4/20 0.57
CDK2 P24941 3/20 0.57
CCNA2 P20248 3/20 0.57
CIT O14578 1/20 0.57
GAK O14976 1/20 0.57
DYRK3 O43781 1/20 0.57
CCNT1 O60563 1/20 0.57
STK16 O75716 1/20 0.57
CCNK O75909 1/20 0.57
STK10 O94804 1/20 0.57
PRKD3 O94806 1/20 0.57
ABCB11 O95342 1/20 0.57
MAP4K4 O95819 1/20 0.57
CCNE2 O96020 1/20 0.57
EGFR P00533 1/20 0.57
NTRK1 P04629 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22650614 0.87 CDK6 (0.75) CDK6CDK4CCND1CDK1CCND3
SCHEMBL19209873 0.83 CDK6 (0.61) CDK6CDK4CCND1CDK1CCND3
SCHEMBL19209865 0.83 CDK6 (0.61) CDK6CDK4CCND1CDK1CCND3
SCHEMBL19231758 0.80 CDK6 (0.53) CDK6CDK4CCND1CDK1CCND3
SCHEMBL17477131 0.78 CDK4 (0.78) CDK6CDK4CCND1CDK1CCND3
SCHEMBL17488748 0.78 CDK4 (0.77) CDK6CDK4CCND1CDK1CCND3
SCHEMBL22650861 0.77 CDK6 (0.50) CDK6CDK4CCND1CDK1CCND3
SCHEMBL21658744 0.77 CDK4 (0.76) CDK6CDK4CCND1CDK1CCND3
SCHEMBL17488745 0.77 CDK4 (0.88) CDK6CDK4CCND1CDK1CCND3
SCHEMBL17489052 0.77 CDK4 (0.88) CDK6CDK4CCND1CDK1CCND3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020224568-A1 CDK INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2020-11-12 WO disclosed