SCHEMBL22650796

SCHEMBL22650796

CC(C)c1cnn2ccc(-c3ccnc(Nc4ccc(C(=O)N5CC(O)C5)cc4)n3)cc12

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 6/20 0.44
CDK1 P06493 5/20 0.44
ACVR1 Q04771 1/20 0.42
MYLK4 Q86YV6 2/20 0.42
STK17A Q9UEE5 2/20 0.42
NEK3 P51956 1/20 0.42
LIMK1 P53667 1/20 0.42
NEK5 Q6P3R8 1/20 0.42
MTOR P42345 1/20 0.41
SMG1 Q96Q15 1/20 0.41
CDK4 P11802 1/20 0.41
CCNB1 P14635 1/20 0.41
CCND1 P24385 1/20 0.41
BTK Q06187 2/20 0.40
IKBKB O14920 3/20 0.40
CHUK O15111 3/20 0.40
IKBKG Q9Y6K9 3/20 0.40
KCNH2 Q12809 2/20 0.39
JAK2 O60674 1/20 0.39
JAK3 P52333 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22650848 0.94 CDK1 (0.49) CDK2CDK1ACVR1MYLK4STK17A
SCHEMBL22650849 0.93 CDK1 (0.47) CDK2CDK1MYLK4STK17ANEK3
SCHEMBL22650927 0.92 CDK2 (0.52) CDK2CDK1ACVR1MYLK4STK17A
SCHEMBL22650800 0.91 IKBKB (0.46) CDK2CDK1ACVR1MYLK4STK17A
SCHEMBL22650921 0.90 MTOR (0.49) CDK2CDK1MYLK4STK17ANEK3
SCHEMBL22650925 0.88 CDK2 (0.61) CDK2CDK1ACVR1MYLK4STK17A
SCHEMBL22650395 0.87 CDK1 (0.61) CDK2CDK1ACVR1MYLK4STK17A
SCHEMBL22650853 0.87 CDK1 (0.52) CDK2CDK1MYLK4STK17ANEK3
SCHEMBL22650851 0.87 IKBKB (0.56) CDK2CDK1MYLK4STK17ANEK3
SCHEMBL22650923 0.85 MAPK8 (0.54) CDK2CDK1ACVR1MYLK4STK17A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020224568-A1 CDK INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2020-11-12 WO disclosed