SCHEMBL22650923

SCHEMBL22650923

CC(C)c1cnn2ccc(-c3ccnc(Nc4ccc(C(N)=O)cc4)n3)cc12

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK8 P45983 4/20 0.54
MAPK10 P53779 1/20 0.54
CDK2 P24941 4/20 0.53
KCNH2 Q12809 2/20 0.53
GSK3B P49841 3/20 0.51
CDK4 P11802 2/20 0.51
JAK2 O60674 1/20 0.48
CAMKK2 Q96RR4 6/20 0.47
PIK3CG P48736 3/20 0.47
IKBKB O14920 2/20 0.45
CHUK O15111 1/20 0.45
ACVR1 Q04771 1/20 0.45
CDK1 P06493 1/20 0.44
CCNB1 P14635 1/20 0.44
CCND1 P24385 1/20 0.44
MYLK4 Q86YV6 2/20 0.44
STK17A Q9UEE5 2/20 0.44
NEK3 P51956 1/20 0.44
LIMK1 P53667 1/20 0.44
NEK5 Q6P3R8 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22650920 0.90 CDK2 (0.54) MAPK8MAPK10CDK2KCNH2CDK4
SCHEMBL22650919 0.89 CDK2 (0.54) MAPK8MAPK10CDK2KCNH2GSK3B
SCHEMBL22650921 0.87 MTOR (0.49) CDK2CDK4IKBKBCHUKCDK1
SCHEMBL22650796 0.85 CDK2 (0.44) CDK2KCNH2CDK4JAK2IKBKB
SCHEMBL22650918 0.85 DKK1 (0.57) MAPK8MAPK10CDK2GSK3BJAK2
SCHEMBL22650849 0.85 CDK1 (0.47) CDK2JAK2IKBKBCHUKCDK1
SCHEMBL22650927 0.84 CDK2 (0.52) CDK2KCNH2CDK4IKBKBCHUK
SCHEMBL22650800 0.83 IKBKB (0.46) CDK2KCNH2CDK4JAK2IKBKB
SCHEMBL22650848 0.83 CDK1 (0.49) CDK2JAK2IKBKBCHUKACVR1
SCHEMBL22650851 0.82 IKBKB (0.56) CDK2IKBKBCHUKCDK1MYLK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020224568-A1 CDK INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2020-11-12 WO disclosed