SCHEMBL22650854

SCHEMBL22650854

CC(C)c1cnn2ccc(-c3ccnc(Nc4ccc(C(=O)N5CCC(N(C)C)C5)cc4F)n3)cc12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 5/20 0.43
CDK1 P06493 4/20 0.43
CDK6 Q00534 2/20 0.42
CDK4 P11802 1/20 0.42
CDK5 Q00535 1/20 0.42
IKBKB O14920 1/20 0.40
CHUK O15111 1/20 0.40
IKBKG Q9Y6K9 1/20 0.40
ATR Q13535 3/20 0.40
LRRK2 Q5S007 2/20 0.40
ABL1 P00519 6/20 0.39
PDGFRB P09619 3/20 0.39
KIT P10721 2/20 0.39
LYN P07948 3/20 0.39
BCR P11274 2/20 0.39
RIPK2 O43353 1/20 0.39
LCK P06239 1/20 0.39
FYN P06241 1/20 0.39
RET P07949 1/20 0.39
ARAF P10398 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22650853 0.89 CDK1 (0.52) CDK2CDK1IKBKBCHUKIKBKG
SCHEMBL22650851 0.85 IKBKB (0.56) CDK2CDK1CDK6IKBKBCHUK
SCHEMBL22650800 0.83 IKBKB (0.46) CDK2CDK1CDK6CDK4IKBKB
SCHEMBL22650597 0.81 EGFR (0.37) CDK2CDK4EGFR
SCHEMBL22650848 0.80 CDK1 (0.49) CDK2CDK1IKBKBCHUKIKBKG
SCHEMBL22650849 0.79 CDK1 (0.47) CDK2CDK1IKBKBCHUKIKBKG
SCHEMBL22650925 0.79 CDK2 (0.61) CDK2CDK1IKBKBCHUKIKBKG
SCHEMBL22650395 0.78 CDK1 (0.61) CDK2CDK1IKBKBCHUKIKBKG
SCHEMBL22650796 0.76 CDK2 (0.44) CDK2CDK1CDK4IKBKBCHUK
SCHEMBL22650921 0.76 MTOR (0.49) CDK2CDK1CDK6CDK4IKBKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020224568-A1 CDK INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2020-11-12 WO disclosed