SCHEMBL22666388

SCHEMBL22666388

Cc1ncc(OC[C@@]2(c3cccc(F)c3)CC2C(=O)O)c(C)n1

nearest known ligand 0.74

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 20/20 0.74
HCRTR2 O43614 20/20 0.74
KCNH2 Q12809 5/20 0.74

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29521524 1.00 HCRTR1 (0.74) HCRTR1HCRTR2KCNH2
SCHEMBL24533939 1.00 HCRTR1 (0.74) HCRTR1HCRTR2KCNH2
SCHEMBL2116763 1.00 HCRTR1 (0.74) HCRTR1HCRTR2KCNH2
SCHEMBL26350991 0.92 HCRTR1 (0.74) HCRTR1HCRTR2KCNH2
SCHEMBL16638936 0.92 HCRTR1 (0.74) HCRTR1HCRTR2KCNH2
SCHEMBL26350983 0.92 HCRTR1 (0.74) HCRTR1HCRTR2KCNH2
SCHEMBL2610558 0.92 HCRTR1 (0.74) HCRTR1HCRTR2KCNH2
SCHEMBL26351279 0.92 HCRTR1 (0.74) HCRTR1HCRTR2KCNH2
SCHEMBL26350998 0.91 HCRTR1 (0.73) HCRTR1HCRTR2KCNH2
SCHEMBL28928604 0.90 HCRTR1 (0.75) HCRTR1HCRTR2KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023178702-A1 METHOD FOR PREPARING LEMBOREXANT AND METHOD FOR PREPARING LEMBOREXANT INTERMEDIATE COMPOUND 浙江华海药业股份有限公司 2023-09-28 WO disclosed
CN-114901285-A Raw material medicine of Leboraseng and medicine composition containing same 卫材R&D管理有限公司 2022-08-12 CN disclosed
WO-2020230800-A1 METHOD AND COMPOUND USEFUL IN PREPARATION OF OREXIN-2 RECEPTOR ANTAGONIST, AND LEMBOREXANT HAVING FEW IMPURITIES エーザイ・アール・アンド・ディー・マネジメント株式会社 2020-11-19 WO disclosed