SCHEMBL22667392

SCHEMBL22667392

COc1cc(O)c2c(=O)cc(-c3ccc(F)cc3)oc2c1N1CCCC1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCNT1 O60563 3/20 0.64
CCNA2 P20248 3/20 0.64
CDK2 P24941 3/20 0.64
CDK9 P50750 3/20 0.64
CDK4 P11802 2/20 0.64
CCND1 P24385 2/20 0.64
CDK7 P50613 2/20 0.64
CCNH P51946 2/20 0.64
MNAT1 P51948 2/20 0.64
CDK6 Q00534 2/20 0.64
USP8 P40818 6/20 0.60
APP P05067 3/20 0.56
ACHE P22303 1/20 0.53
PLK1 P53350 1/20 0.53
BACE1 P56817 1/20 0.53
AR P10275 1/20 0.51
CYP1A1 P04798 1/20 0.50
CYP1A2 P05177 1/20 0.50
CYP1B1 Q16678 1/20 0.50
PARP1 P09874 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29877108 0.90 CYP1A1 (0.56) CCNT1CCNA2CDK2CDK9CDK4
SCHEMBL22667393 0.90 CYP1A1 (0.56) CCNT1CCNA2CDK2CDK9CDK4
SCHEMBL28848637 0.87 USP8 (0.58) CCNT1CCNA2CDK2CDK9CDK4
SCHEMBL22667394 0.86 CCNT1 (0.84) CCNT1CCNA2CDK2CDK9CDK4
SCHEMBL22667441 0.85 CCNT1 (0.83) CCNT1CCNA2CDK2CDK9CDK4
SCHEMBL22667227 0.82 CCNT1 (0.91) CCNT1CCNA2CDK2CDK9CDK4
SCHEMBL22667374 0.79 CCNT1 (0.83) CCNT1CCNA2CDK2CDK9CDK4
SCHEMBL22667228 0.79 CCNT1 (0.85) CCNT1CCNA2CDK2CDK9CDK4
SCHEMBL22667451 0.78 CCNT1 (0.80) CCNT1CCNA2CDK2CDK9CDK4
SCHEMBL22667258 0.78 CCNT1 (1.00) CCNT1CCNA2CDK2CDK9CDK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114957182-B USP8 inhibitor containing flavone skeleton structure and application thereof 中国药科大学 2024-03-15 CN disclosed
CN-114957182-A USP8 inhibitor containing flavone skeleton structure and application thereof 中国药科大学 2022-08-30 CN disclosed
WO-2020228513-A1 NOVEL CDK9 INHIBITOR BASED ON BENZOPYRAN STRUCTURE, PREPARATION METHOD THEREFOR AND USE THEREOF 中国药科大学 2020-11-19 WO disclosed