SCHEMBL22682013

SCHEMBL22682013

COc1ccccc1-c1ccc2c(c1)OCCC2

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTNNB1 P35222 1/20 0.53
WNT3A P56704 1/20 0.53
PTPRC P08575 1/20 0.44
PTPN1 P18031 1/20 0.44
CTSG P08311 2/20 0.43
KLK7 P49862 2/20 0.43
KLK14 Q9P0G3 2/20 0.43
KLK5 Q9Y337 2/20 0.43
PDGFRB P09619 1/20 0.43
FGFR1 P11362 1/20 0.43
KDR P35968 1/20 0.43
KDM4C Q9H3R0 1/20 0.41
PDK2 Q15119 1/20 0.41
DHFR P00374 1/20 0.41
ADORA1 P30542 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
KCNH2 Q12809 1/20 0.40
HSD17B3 P37058 1/20 0.40
MEN1 O00255 1/20 0.40
ALDH1A1 P00352 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22681887 0.85 BACE1 (0.51) CTNNB1WNT3AKDM4CKCNH2LMNA
SCHEMBL17378737 0.85 CTNNB1 (0.45) CTNNB1WNT3AKDM4CKCNH2ESR1
SCHEMBL22681889 0.81 CD274 (0.42) CTNNB1WNT3AKDM4CPDK2ADORA1
SCHEMBL6951619 0.79 ADORA1 (0.52) PTPRCPTPN1PDGFRBFGFR1KDR
SCHEMBL22681721 0.78 MEN1 (0.44) CTNNB1WNT3AKDM4CKCNH2MEN1
SCHEMBL22681646 0.78 AXL (0.47) CTSGKLK7KLK14KLK5KDM4C
SCHEMBL28137011 0.76 KCNH2 (0.52) CTNNB1WNT3AKCNH2
SCHEMBL22681657 0.75 CTNNB1 (0.45) CTNNB1WNT3AKDM4CKCNH2ALDH1A1
SCHEMBL22681716 0.75 ESR2 (0.43) KDM4CKCNH2HSD17B3MEN1ALDH1A1
SCHEMBL22681979 0.75 KCNH2 (0.44) CTNNB1WNT3AKDM4CKCNH2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3160952-B1 HISTONE DEMETHYLASE INHIBITORS CELGENE QUANTICEL RES INC (US) 2020-12-02 EP disclosed
EP-3741749-A1 HISTONE DEMETHYLASE INHIBITORS Celgene Quanticel Research, Inc. (US) 2020-11-25 EP disclosed
EP-3738960-A1 HISTONE DEMETHYLASE INHIBITORS Celgene Quanticel Research, Inc. (US) 2020-11-18 EP disclosed