SCHEMBL22685276

SCHEMBL22685276

Cc1cc(=O)[nH]c(=O)n1N

nearest known ligand 0.44

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.44
KDM4E B2RXH2 2/20 0.44
GAA P10253 2/20 0.44
TYMP P19971 13/20 0.43
ATM Q13315 1/20 0.43
CRBN Q96SW2 1/20 0.40
CA1 P00915 1/20 0.38
LMNA P02545 1/20 0.38
MEN1 O00255 1/20 0.38
GLA P06280 1/20 0.38
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6027678 0.76 TYMP (0.46) ALDH1A1KDM4EGAATYMPATM
SCHEMBL28263643 0.73 TYMP (0.43) ALDH1A1KDM4EGAATYMPATM
SCHEMBL27816353 0.73 TYMP (0.45) ALDH1A1KDM4EGAATYMPATM
SCHEMBL4960409 0.70 POLB (0.46) ALDH1A1KDM4EGAATYMPATM
SCHEMBL12702529 0.70 TYMP (0.41) ALDH1A1KDM4EGAATYMPATM
SCHEMBL15469004 0.70 POLB (0.43) ALDH1A1KDM4EGAATYMPATM
SCHEMBL8768819 0.68 TYMP (0.44) ALDH1A1KDM4ETYMPATMMEN1
SCHEMBL9191218 0.68 ATM (0.44) ALDH1A1KDM4EGAATYMPATM
SCHEMBL30493068 0.68 CRBN (0.36) ALDH1A1KDM4EGAACRBNLMNA
SCHEMBL4469664 0.67 KDM4E (0.45) ALDH1A1KDM4EGAATYMPATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3795568-A1 FLUORINATED LYSYL OXIDASE-LIKE 2 INHIBITORS AND USES THEREOF Pharmakea, Inc. (US) 2021-03-24 EP disclosed
EP-3265456-B1 FLUORINATED LYSYL OXIDASE-LIKE 2 INHIBITORS AND USES THEREOF PHARMAKEA INC (US) 2020-11-18 EP disclosed