SCHEMBL2268792

SCHEMBL2268792

O=C(NCc1ccc2c(c1)CCN(C1CCC1)CC2)c1cnc(N2CCC(F)(F)C2)cn1

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 13/20 0.47
CACNA1G O43497 1/20 0.46
CACNA1H O95180 1/20 0.46
CACNA1I Q9P0X4 1/20 0.46
HRH1 P35367 1/20 0.46
KLKB1 P03952 4/20 0.41
KLK1 P06870 2/20 0.41
PRKAB2 O43741 1/20 0.37
PRKAG1 P54619 1/20 0.37
PRKAA2 P54646 1/20 0.37
PRKAA1 Q13131 1/20 0.37
PRKAG3 Q9UGI9 1/20 0.37
PRKAG2 Q9UGJ0 1/20 0.37
PRKAB1 Q9Y478 1/20 0.37
NAPEPLD Q6IQ20 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6860616 0.89 HRH3 (0.49) HRH3CACNA1GCACNA1HCACNA1IHRH1
SCHEMBL2270394 0.86 HRH3 (0.49) HRH3HRH1KLKB1KLK1
SCHEMBL2347977 0.86 HRH3 (0.49) HRH3HRH1KLKB1KLK1
SCHEMBL2193364 0.86 HRH3 (0.45) HRH3CACNA1GCACNA1HCACNA1IHRH1
SCHEMBL2365248 0.86 HRH3 (0.49) HRH3HRH1KLKB1KLK1
SCHEMBL2271409 0.85 HRH3 (0.50) HRH3CACNA1GCACNA1HCACNA1IHRH1
SCHEMBL2193394 0.83 HRH3 (0.45) HRH3HRH1PRKAB2PRKAG1PRKAA2
SCHEMBL2266847 0.81 HRH3 (0.50) HRH3HRH1KLKB1KLK1NAPEPLD
SCHEMBL2269495 0.81 HRH3 (0.50) HRH3HRH1KLKB1KLK1NAPEPLD
SCHEMBL2275230 0.81 HRH3 (0.55) HRH3HRH1PRKAB2PRKAG1PRKAA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011083315-A1 COMPOUNDS AND THEIR USE TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2011-07-14 WO claimed
WO-2011083315-A1 COMPOUNDS AND THEIR USE TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2011-07-14 WO disclosed
WO-2011083315-A1 COMPOUNDS AND THEIR USE TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2011-07-14 WO disclosed