SCHEMBL2365248

SCHEMBL2365248

O=C(NCc1ccc2c(c1)CCN(C1CCC1)CC2)c1cnc(N2CCC(F)C2)cn1

nearest known ligand 0.49

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 13/20 0.49
HRH1 P35367 1/20 0.47
KLKB1 P03952 4/20 0.41
KLK1 P06870 2/20 0.41
ADRA2C P18825 1/20 0.38
CYP2D6 P10635 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2347977 1.00 HRH3 (0.49) HRH3HRH1KLKB1KLK1ADRA2C
SCHEMBL2270394 1.00 HRH3 (0.49) HRH3HRH1KLKB1KLK1ADRA2C
SCHEMBL2266847 0.88 HRH3 (0.50) HRH3HRH1KLKB1KLK1CYP2D6
SCHEMBL2269495 0.88 HRH3 (0.50) HRH3HRH1KLKB1KLK1CYP2D6
SCHEMBL1787838 0.88 HRH3 (0.49) HRH3KLKB1KLK1
SCHEMBL1788393 0.88 HRH3 (0.49) HRH3KLKB1KLK1
SCHEMBL1787839 0.88 HRH3 (0.49) HRH3KLKB1KLK1
SCHEMBL2268792 0.86 HRH3 (0.47) HRH3HRH1KLKB1KLK1
SCHEMBL1787502 0.84 HRH3 (0.45) HRH3HRH1KLKB1KLK1
SCHEMBL1788640 0.84 HRH3 (0.45) HRH3HRH1KLKB1KLK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011083315-A1 COMPOUNDS AND THEIR USE TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2011-07-14 WO disclosed