SCHEMBL22700147

SCHEMBL22700147

CCOP(=O)(OCC)OC[C@H]1O[C@@H](n2cnc3c(N)nc(Cl)nc32)C(C)(COCc2ccccc2)C1O

nearest known ligand 0.53

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PDE2A O00408 4/20 0.53
NT5E P21589 10/20 0.50
ADORA2A P29274 1/20 0.50
ADORA3 P0DMS8 1/20 0.47
P2RY1 P47900 4/20 0.46
P2RY11 Q96G91 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19974455 1.00 PDE2A (0.53) PDE2ANT5EADORA2AADORA3P2RY1
SCHEMBL19974411 0.89 PDE2A (0.46) PDE2ANT5EADORA2AADORA3
SCHEMBL22700164 0.87 PDE2A (0.52) PDE2ANT5EADORA3P2RY1P2RY11
SCHEMBL19979029 0.87 ADORA2A (0.57) NT5EADORA2AADORA3P2RY1P2RY11
SCHEMBL19974418 0.87 ADORA2A (0.57) NT5EADORA2AADORA3P2RY1P2RY11
SCHEMBL19974427 0.86 ADORA2A (0.68) PDE2ANT5EADORA2AADORA3
SCHEMBL19975000 0.80 ADORA2A (0.58) NT5EADORA2AADORA3P2RY1P2RY11
SCHEMBL22700162 0.79 PDE2A (0.46) PDE2ANT5EADORA3
SCHEMBL19974603 0.78 NT5E (0.44) NT5EADORA2AADORA3P2RY1P2RY11
SCHEMBL19974435 0.78 ADORA2A (0.49) NT5EADORA2AADORA3P2RY1P2RY11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3512860-B1 NUCLEOSIDE AND NUCLEOTIDE ANALOGUES BEARING A QUATERNARY ALL-CARBON STEREOGENIC CENTER AT THE 2' POSITION AND METHODS OF USE AS A CARDIOPROTECTIVE AGENT LCB PHARMA INC (CA) 2020-11-25 EP disclosed