SCHEMBL22701124

SCHEMBL22701124

C=Nc1ncnc2[nH]ccc(=O)c12

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.35
RAB9A P51151 2/20 0.34
KMT2A Q03164 2/20 0.34
ALDH1A1 P00352 1/20 0.34
GLA P06280 1/20 0.34
POLB P06746 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
CCNT1 O60563 2/20 0.33
CCNA2 P20248 2/20 0.33
CDK2 P24941 2/20 0.33
CDK9 P50750 2/20 0.33
CCNA1 P78396 2/20 0.33
CDK5 Q00535 2/20 0.33
CDK5R1 Q15078 2/20 0.33
ADORA2A P29274 1/20 0.33
ADORA1 P30542 1/20 0.33
JAK2 O60674 2/20 0.33
JAK1 P23458 2/20 0.31
NOTUM Q6P988 1/20 0.31
IKBKB O14920 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1599110 0.75 KDM4E (0.38) KDM4ERAB9AKMT2AALDH1A1GLA
SCHEMBL15086999 0.75 JAK2 (0.47) JAK2JAK1NOTUMIKBKBCHUK
SCHEMBL3767011 0.74 KDM4E (0.37) KDM4ERAB9AKMT2AALDH1A1GLA
SCHEMBL19153637 0.74 KDM4E (0.51) KDM4ERAB9AKMT2AALDH1A1GLA
SCHEMBL6833739 0.74 CHEK1 (0.49) KDM4ERAB9AKMT2AALDH1A1GLA
SCHEMBL12391478 0.71 LRRK2 (0.40) KDM4ERAB9AKMT2AALDH1A1GLA
SCHEMBL21388537 0.70 JAK3 (0.40) KDM4ERAB9AKMT2AALDH1A1GLA
SCHEMBL18238494 0.70 ADORA2A (0.40) KDM4ERAB9AKMT2AALDH1A1GLA
SCHEMBL3761579 0.67 TTBK1 (0.55) JAK2JAK1TTBK1TTBK2
SCHEMBL13058088 0.66 TTBK1 (0.45) JAK2JAK1TTBK1TTBK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020234756-A1 PYRIDO-PYRIMIDIN DERIVATIVES AND PHARMACEUTICAL COMPOSITION, FOR USE IN PREVENTING OR TREATING PI3 KINASE RELATED DISEASES, COMPRISING SAME AS ACTIVE INGREDIENT 보령제약 주식회사 (KR) 2020-11-26 WO disclosed