SCHEMBL22701997

SCHEMBL22701997

O=C(O)/C=C/[S+]([O-])c1ccc2ccccc2c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TBXA2R P21731 1/20 0.40
PTGER4 P35408 1/20 0.40
PTGFR P43088 1/20 0.40
PTGER3 P43115 1/20 0.40
PTGER2 P43116 1/20 0.40
PTGDR Q13258 1/20 0.40
CYP1B1 Q16678 1/20 0.40
ESR1 P03372 1/20 0.39
CCNC P24863 1/20 0.38
CDK8 P49336 1/20 0.38
CES2 O00748 1/20 0.38
CES1 P23141 1/20 0.38
KDM4E B2RXH2 2/20 0.37
LMNA P02545 1/20 0.37
MAPT P10636 3/20 0.37
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
TDP1 Q9NUW8 2/20 0.37
ALDH1A1 P00352 1/20 0.37
EGFR P00533 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19235254 0.82 CCNC (0.43) CCNCCDK8KDM4EMAPTMEN1
SCHEMBL9330870 0.81 HCAR2 (0.43) KDM4ELMNAMAPTMEN1KMT2A
SCHEMBL9845559 0.81 HCAR2 (0.43) KDM4ELMNAMAPTMEN1KMT2A
SCHEMBL9845672 0.81 HCAR2 (0.43) KDM4ELMNAMAPTMEN1KMT2A
SCHEMBL7928592 0.74 PTGER3 (0.50) TBXA2RPTGER4PTGFRPTGER3PTGER2
SCHEMBL7824273 0.74 PTGER3 (0.50) TBXA2RPTGER4PTGFRPTGER3PTGER2
SCHEMBL11371545 0.70 PTPN7 (0.45) CES2CES1MAPTMEN1KMT2A
Naphthalene SCHEMBL2834571 0.70 HCAR2 (0.56) KDM4ELMNAMAPTKMT2AALDH1A1
Naphthalene SCHEMBL2834576 0.70 HCAR2 (0.56) KDM4ELMNAMAPTKMT2AALDH1A1
SCHEMBL238071 0.69 CYP2A6 (0.39) ESR1CES2CES1LMNATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3411361-B1 NRF2 ACTIVATING COMPOUNDS AND USES THEREOF RIGEL PHARMACEUTICALS INC (US) 2020-11-25 EP disclosed